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2R40

Crystal structure of 20E bound EcR/USP

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0003707molecular_functionnuclear steroid receptor activity
A0005515molecular_functionprotein binding
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
A0008270molecular_functionzinc ion binding
A0030518biological_processnuclear receptor-mediated steroid hormone signaling pathway
D0003677molecular_functionDNA binding
D0004879molecular_functionnuclear receptor activity
D0005634cellular_componentnucleus
D0006355biological_processregulation of DNA-templated transcription
D0035076biological_processecdysone receptor signaling pathway
D0035100molecular_functionecdysone binding
Functional Information from PDB Data
site_idAC1
Number of Residues2
DetailsBINDING SITE FOR RESIDUE FLC D 9400
ChainResidue
DGLY359
DTYR464

site_idAC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 D 1327
ChainResidue
DTHR291
DASN293
DTYR464

site_idAC3
Number of Residues17
DetailsBINDING SITE FOR RESIDUE 20E D 9001
ChainResidue
DTHR346
DMET380
DARG383
DARG387
DLEU396
DPHE397
DALA398
DTYR408
DVAL416
DLEU420
DASN504
DTRP526
DHOH9517
DGLU309
DGLN310
DMET342
DTHR343

site_idAC4
Number of Residues16
DetailsBINDING SITE FOR RESIDUE EPH A 600
ChainResidue
AVAL238
APRO239
APHE242
ALEU249
AASN287
ALEU291
ASER335
AGLN338
AALA339
AGLY340
AVAL341
APHE345
ASER431
AHIS434
AHOH613
AHOH624

site_idAC5
Number of Residues1
DetailsBINDING SITE FOR RESIDUE GOL D 9500
ChainResidue
DHOH9544

238895

PDB entries from 2025-07-16

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