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2QJ4

A Mechanistic Basis for Converting a Receptor Tyrosine Kinase Agonist to an Antagonist

Functional Information from PDB Data
site_idAC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 3001
ChainResidue
ALYS61
ATHR62
BLYS64
BARG94
BARG96

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 3002
ChainResidue
BTHR62
BHOH2034
ALYS64
AARG94
AARG96
BLYS61

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 3003
ChainResidue
ALYS63
ALYS64
AARG96
BLYS63
BLYS64
BARG96

Functional Information from PROSITE/UniProt
site_idPS00021
Number of Residues14
DetailsKRINGLE_1 Kringle domain signature. YCRNprgeeggpWC
ChainResidueDetails
ATYR177-CYS190

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues156
DetailsDomain: {"description":"Kringle 1","evidences":[{"source":"PROSITE-ProRule","id":"PRU00121","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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