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2QJ2

A Mechanistic Basis for Converting a Receptor Tyrosine Kinase Agonist to an Antagonist

Functional Information from PDB Data
site_idAC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 3001
ChainResidue
ALYS60
ALYS62
AARG73
ATYR167
AARG181

site_idAC2
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 A 3002
ChainResidue
AARG134
ASER135
ATYR136
AHOH2217
AARG126
AILE130
AGLY131
AGLY133

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 B 3003
ChainResidue
BHIS1160
BSER1161
BPHE1162
BARG1168
BARG1197
BHOH2228
BHOH2303

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 3004
ChainResidue
AARG168
AGLY169
AASP171
AHOH2027
AHOH2278

Functional Information from PROSITE/UniProt
site_idPS00021
Number of Residues14
DetailsKRINGLE_1 Kringle domain signature. YCRNprgeeggpWC
ChainResidueDetails
ATYR176-CYS189

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Pyrrolidone carboxylic acid => ECO:0000269|PubMed:1826837
ChainResidueDetails
AGLN32
BGLN1032

222926

PDB entries from 2024-07-24

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