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2O9I

Crystal Structure of the Human Pregnane X Receptor LBD in complex with an SRC-1 coactivator peptide and T0901317

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues15
DetailsBINDING SITE FOR RESIDUE 444 B 1
ChainResidue
BLEU1206
BLEU1324
BHIS1327
BHIS1407
BLEU1411
BILE1414
BPHE1420
BLEU1209
BMET1243
BSER1247
BGLN1285
BPHE1288
BTRP1299
BTYR1306
BMET1323

site_idAC2
Number of Residues15
DetailsBINDING SITE FOR RESIDUE 444 A 2
ChainResidue
ALEU209
AVAL211
ALEU240
AMET243
AMET246
AGLN285
APHE288
ATRP299
ATYR306
ALEU308
AHIS327
AHIS407
ALEU411
APHE420
AMET425

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues10
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"12578355","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1M13","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 4"}
ChainResidueDetails

239149

PDB entries from 2025-07-23

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