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2JF9

ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH A TAMOXIFEN-SPECIFIC PEPTIDE ANTAGONIST

Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE BCT A 700
ChainResidue
ALEU327
ATYR328
AARG352
CILE326
CLEU327
CTYR328
CARG352

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CA P 1014
ChainResidue
PASP10
PSER13
CTHR334
CHOH2021

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CA R 1014
ChainResidue
ATHR334
AHOH2018
RASP10
RSER13

site_idAC4
Number of Residues16
DetailsBINDING SITE FOR RESIDUE OHT A 600
ChainResidue
AMET343
ALEU346
ATHR347
AALA350
AASP351
AGLU353
ATRP383
ALEU384
AARG394
APHE404
AMET421
ALEU428
AGLY521
AHIS524
ALEU525
PPRO2

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1529
ChainResidue
ATYR331
APRO333
AASN407
AHOH2095
CASN359

site_idAC6
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 1530
ChainResidue
AGLU323
ATRP393
AGLY442
AHOH2096

site_idAC7
Number of Residues13
DetailsBINDING SITE FOR RESIDUE OHT B 600
ChainResidue
BMET343
BLEU346
BTHR347
BALA350
BASP351
BGLU353
BLEU384
BARG394
BPHE404
BMET421
BLEU428
BGLY521
QPRO2

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO B 1530
ChainResidue
ATYR459
BMET427
BTHR431
BHIS513
BHIS516

site_idAC9
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO B 1531
ChainResidue
BLEU320
BGLU323
BTRP393
BGLY442

site_idBC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE OHT C 600
ChainResidue
CMET343
CLEU346
CALA350
CASP351
CGLU353
CARG394
CMET421
CILE424
CLEU428
CHIS524
CLEU525
RSER1
RPRO2

site_idBC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO C 1530
ChainResidue
AVAL355
AASN359
CTYR331
CASN407

site_idBC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO C 1531
ChainResidue
CLEU320
CGLU323
CTRP393
CGLY442

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
ACYS447
BCYS447
CCYS447

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PDB entries from 2024-07-24

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