1SJ0
Human Estrogen Receptor Alpha Ligand-binding Domain in Complex with the Antagonist Ligand 4-D
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 14 |
Details | BINDING SITE FOR RESIDUE E4D A 600 |
Chain | Residue |
A | MET343 |
A | GLY521 |
A | HIS524 |
A | LEU525 |
A | CYS530 |
A | HOH1005 |
A | LEU346 |
A | ALA350 |
A | ASP351 |
A | GLU353 |
A | LEU354 |
A | TRP383 |
A | LEU387 |
A | ARG394 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 3 |
Details | BINDING: BINDING => ECO:0000269|PubMed:9338790, ECO:0000269|PubMed:9600906, ECO:0007744|PDB:1A52, ECO:0007744|PDB:1ERE |
Chain | Residue | Details |
A | GLU353 | |
A | ARG394 | |
A | HIS524 |
site_id | SWS_FT_FI2 |
Number of Residues | 1 |
Details | MOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106 |
Chain | Residue | Details |
A | TYR537 |
site_id | SWS_FT_FI3 |
Number of Residues | 1 |
Details | LIPID: S-palmitoyl cysteine => ECO:0000250 |
Chain | Residue | Details |
A | CYS447 |