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1R4I

Crystal Structure of Androgen Receptor DNA-Binding Domain Bound to a Direct Repeat Response Element

Functional Information from GO Data
ChainGOidnamespacecontents
A0003700molecular_functionDNA-binding transcription factor activity
A0006355biological_processregulation of DNA-templated transcription
A0008270molecular_functionzinc ion binding
A0043565molecular_functionsequence-specific DNA binding
B0003700molecular_functionDNA-binding transcription factor activity
B0006355biological_processregulation of DNA-templated transcription
B0008270molecular_functionzinc ion binding
B0043565molecular_functionsequence-specific DNA binding
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 650
ChainResidue
ACYS542
ACYS545
ACYS559
ACYS562

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 651
ChainResidue
ACYS578
ACYS584
ACYS594
ACYS597

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN B 652
ChainResidue
BCYS545
BCYS559
BCYS562
BCYS542

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN B 653
ChainResidue
BCYS578
BCYS584
BCYS594
BCYS597

Functional Information from PROSITE/UniProt
site_idPS00031
Number of Residues27
DetailsNUCLEAR_REC_DBD_1 Nuclear hormones receptors DNA-binding region signature. CliCg.Deasga.HYgaltCgsCkvFFkR
ChainResidueDetails
ACYS542-ARG568

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues146
DetailsDNA_BIND: Nuclear receptor => ECO:0000255|PROSITE-ProRule:PRU00407
ChainResidueDetails
ATHR541-LEU614
BTHR541-LEU614

site_idSWS_FT_FI2
Number of Residues88
DetailsZN_FING: NR C4-type => ECO:0000255|PROSITE-ProRule:PRU00407
ChainResidueDetails
ACYS542-CYS562
ACYS578-CYS602
BCYS542-CYS562
BCYS578-CYS602

site_idSWS_FT_FI3
Number of Residues2
DetailsMOD_RES: Phosphotyrosine; by CSK => ECO:0000250|UniProtKB:P10275
ChainResidueDetails
ATYR534
BTYR534

site_idSWS_FT_FI4
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:22673903
ChainResidueDetails
ASER633
BSER633

218853

PDB entries from 2024-04-24

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