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1O0K

Structure of the First Parallel DNA Quadruplex-drug Complex

Functional Information from PDB Data
site_id1
Number of Residues
Details
ChainResidue

site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE DM1 B 25
ChainResidue
ADT1001
CDG1015
CDG1016
DDM126
ADT1001
BDG1008
BHOH1107
BHOH1124
BHOH1185
CDM127
CDM127
CDG1014

site_idAC2
Number of Residues12
DetailsBINDING SITE FOR RESIDUE DM1 D 26
ChainResidue
ADG1002
ADG1003
AHOH1116
BDM125
CDM127
CDM127
CDT1013
CDT1018
DDT1019
DDG1020
DHOH1101
DHOH1140

site_idAC3
Number of Residues19
DetailsBINDING SITE FOR RESIDUE DM1 C 27
ChainResidue
ADT1001
BDM125
BDM125
CDT1013
CDG1014
CDT1018
CHOH1106
CHOH1110
CHOH1126
CHOH1128
CHOH1129
CHOH1132
CHOH1134
CHOH1156
CHOH1159
CHOH1200
DDM126
DDM126
DDT1019

site_idAC4
Number of Residues9
DetailsBINDING SITE FOR RESIDUE NA A 28
ChainResidue
ADG1004
ADG1005
BDG1010
BDG1011
CNA29
CDG1016
CDG1017
DDG1022
DDG1023

site_idAC5
Number of Residues10
DetailsBINDING SITE FOR RESIDUE NA C 29
ChainResidue
ANA28
ANA30
ADG1003
ADG1004
BDG1009
BDG1010
CDG1015
CDG1016
DDG1021
DDG1022

site_idAC6
Number of Residues9
DetailsBINDING SITE FOR RESIDUE NA A 30
ChainResidue
ADG1002
ADG1003
BDG1008
BDG1009
CNA29
CDG1014
CDG1015
DDG1020
DDG1021

224572

PDB entries from 2024-09-04

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