1NHG
CRYSTAL STRUCTURE ANALYSIS OF PLASMODIUM FALCIPARUM ENOYL-ACYL-CARRIER-PROTEIN REDUCTASE WITH TRICLOSAN
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0004318 | molecular_function | enoyl-[acyl-carrier-protein] reductase (NADH) activity |
A | 0006633 | biological_process | fatty acid biosynthetic process |
B | 0004318 | molecular_function | enoyl-[acyl-carrier-protein] reductase (NADH) activity |
B | 0006633 | biological_process | fatty acid biosynthetic process |
C | 0004318 | molecular_function | enoyl-[acyl-carrier-protein] reductase (NADH) activity |
C | 0006633 | biological_process | fatty acid biosynthetic process |
D | 0004318 | molecular_function | enoyl-[acyl-carrier-protein] reductase (NADH) activity |
D | 0006633 | biological_process | fatty acid biosynthetic process |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 23 |
Details | BINDING SITE FOR RESIDUE NAD A 450 |
Chain | Residue |
A | GLY104 |
A | SER215 |
A | LEU216 |
A | ALA217 |
A | ASN218 |
A | LEU265 |
A | THR266 |
A | LYS285 |
A | ALA312 |
A | GLY313 |
A | PRO314 |
A | ILE105 |
A | LEU315 |
A | SER317 |
A | ALA319 |
A | TCL500 |
A | GLY106 |
A | GLY110 |
A | TYR111 |
A | TRP131 |
A | PHE167 |
A | ASP168 |
A | ALA169 |
site_id | AC2 |
Number of Residues | 21 |
Details | BINDING SITE FOR RESIDUE NAD B 550 |
Chain | Residue |
B | ILE105 |
B | GLY106 |
B | GLY110 |
B | TYR111 |
B | TRP131 |
B | PHE167 |
B | ASP168 |
B | ALA169 |
B | SER215 |
B | LEU216 |
B | ASN218 |
B | LEU265 |
B | THR266 |
B | LYS285 |
B | ALA312 |
B | GLY313 |
B | PRO314 |
B | LEU315 |
B | SER317 |
B | ALA319 |
B | TCL600 |
site_id | AC3 |
Number of Residues | 9 |
Details | BINDING SITE FOR RESIDUE TCL A 500 |
Chain | Residue |
A | ALA217 |
A | ASN218 |
A | ALA219 |
A | TYR267 |
A | TYR277 |
A | ALA319 |
A | ILE323 |
A | NAD450 |
C | PHE368 |
site_id | AC4 |
Number of Residues | 8 |
Details | BINDING SITE FOR RESIDUE TCL B 600 |
Chain | Residue |
B | ALA217 |
B | ASN218 |
B | ALA219 |
B | TYR267 |
B | TYR277 |
B | ALA319 |
B | NAD550 |
D | PHE368 |
Catalytic Information from CSA
site_id | CSA1 |
Number of Residues | 2 |
Details | Annotated By Reference To The Literature 1qsg |
Chain | Residue | Details |
A | TYR277 | |
A | LYS285 |
site_id | CSA2 |
Number of Residues | 2 |
Details | Annotated By Reference To The Literature 1qsg |
Chain | Residue | Details |
B | TYR277 | |
B | LYS285 |
site_id | CSA3 |
Number of Residues | 2 |
Details | Annotated By Reference To The Literature 1qsg |
Chain | Residue | Details |
A | MET281 | |
A | LYS285 |
site_id | CSA4 |
Number of Residues | 2 |
Details | Annotated By Reference To The Literature 1qsg |
Chain | Residue | Details |
B | MET281 | |
B | LYS285 |