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1KIE

Inosine-adenosine-guanosine preferring nucleoside hydrolase from Trypanosoma vivax: Asp10Ala mutant in complex with 3-deaza-adenosine

Functional Information from GO Data
ChainGOidnamespacecontents
A0005829cellular_componentcytosol
A0006152biological_processpurine nucleoside catabolic process
A0008477molecular_functionpurine nucleosidase activity
A0016799molecular_functionhydrolase activity, hydrolyzing N-glycosyl compounds
B0005829cellular_componentcytosol
B0006152biological_processpurine nucleoside catabolic process
B0008477molecular_functionpurine nucleosidase activity
B0016799molecular_functionhydrolase activity, hydrolyzing N-glycosyl compounds
Functional Information from PDB Data
site_idAC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CA A 328
ChainResidue
AASP15
ATHR137
AASP261
AAD3801
AHOH809

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CA B 328
ChainResidue
BHOH814
BASP15
BTHR137
BASP261
BAD3802

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE NI A 701
ChainResidue
AGLU44
AGLU113
AHOH957

site_idAC4
Number of Residues11
DetailsBINDING SITE FOR RESIDUE AD3 A 801
ChainResidue
AASP14
AASP40
ATHR137
AMET164
AASN173
AGLU184
AASN186
ATRP260
AASP261
ACA328
AHOH809

site_idAC5
Number of Residues14
DetailsBINDING SITE FOR RESIDUE AD3 B 802
ChainResidue
BASN12
BASP14
BASP15
BASP40
BTRP83
BTHR137
BMET164
BASN173
BGLU184
BTRP185
BASN186
BTRP260
BASP261
BCA328

Catalytic Information from CSA
site_idMCSA1
Number of Residues8
DetailsM-CSA 471
ChainResidueDetails
AALA10metal ligand, proton shuttle (general acid/base)
AASP15metal ligand
AASP40activator
ATRP83activator
ATHR137metal ligand
AASN186activator, electrostatic stabiliser
ATRP260activator, electrostatic stabiliser
AASP261metal ligand

site_idMCSA2
Number of Residues8
DetailsM-CSA 471
ChainResidueDetails
BALA10metal ligand, proton shuttle (general acid/base)
BASP15metal ligand
BASP40activator
BTRP83activator
BTHR137metal ligand
BASN186activator, electrostatic stabiliser
BTRP260activator, electrostatic stabiliser
BASP261metal ligand

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PDB entries from 2026-03-25

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