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1IJR

Crystal structure of LCK SH2 complexed with nonpeptide phosphotyrosine mimetic

Functional Information from PDB Data
site_idAC1
Number of Residues15
DetailsBINDING SITE FOR RESIDUE CC0 A 150
ChainResidue
ALEU10
ACYS42
AHIS58
ATYR59
ALYS60
AILE71
AGLY93
AARG12
AASP14
AARG17
AGLN18
AARG32
ASER34
AGLU35
ASER36

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphothreonine => ECO:0007744|PubMed:19690332
ChainResidueDetails
ATHR37

site_idSWS_FT_FI2
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:19690332
ChainResidueDetails
ASER40
ASER72

site_idSWS_FT_FI3
Number of Residues1
DetailsMOD_RES: Phosphotyrosine => ECO:0000250|UniProtKB:P06240
ChainResidueDetails
ATYR70

219869

PDB entries from 2024-05-15

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