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8EX0

Crystal structure of JAK2 JH2 (pseudokinase domain) in complex with CDK2-IV

Experimental procedure
Experimental methodSINGLE WAVELENGTH
Source typeSYNCHROTRON
Source detailsAPS BEAMLINE 19-BM
Synchrotron siteAPS
Beamline19-BM
Temperature [K]100
Detector technologyCCD
Collection date2017-08-18
DetectorADSC QUANTUM 210r
Wavelength(s)0.9794
Spacegroup nameP 1 21 1
Unit cell lengths43.986, 57.576, 61.185
Unit cell angles90.00, 110.38, 90.00
Refinement procedure
Resolution29.030 - 1.850
R-factor0.1792
Rwork0.175
R-free0.22760
Structure solution methodFOURIER SYNTHESIS
RMSD bond length0.011
RMSD bond angle1.048
Data reduction softwareHKL-2000
Data scaling softwareHKL-2000
Phasing softwarePHENIX
Refinement softwarePHENIX (1.20.1_4487)
Data quality characteristics
 OverallOuter shell
Low resolution limit [Å]29.0301.880
High resolution limit [Å]1.8501.850
Rmerge0.0620.598
Number of reflections248531229
<I/σ(I)>13.6
Completeness [%]99.9100
Redundancy3.83.7
CC(1/2)0.858
Crystallization Conditions
crystal IDmethodpHtemperaturedetails
1VAPOR DIFFUSION, HANGING DROP9.5277CHES, PEG 3000

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