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6E3T

Crystal Structure of the Heterodimeric HIF-2 Complex with Antagonist T1001

Experimental procedure
Experimental methodSINGLE WAVELENGTH
Source typeSYNCHROTRON
Source detailsAPS BEAMLINE 19-ID
Synchrotron siteAPS
Beamline19-ID
Temperature [K]100
Detector technologyCCD
Collection date2016-04-16
DetectorADSC QUANTUM 315r
Wavelength(s)0.97929
Spacegroup nameP 1 21 1
Unit cell lengths49.032, 97.981, 77.427
Unit cell angles90.00, 107.10, 90.00
Refinement procedure
Resolution41.793 - 3.000
R-factor0.2485
Rwork0.245
R-free0.30640
Structure solution methodMOLECULAR REPLACEMENT
Starting model (for MR)4zp4
RMSD bond length0.012
RMSD bond angle1.586
Data scaling softwareHKL-3000
Phasing softwarePHASER
Refinement softwarePHENIX ((dev_2467: ???))
Data quality characteristics
 OverallOuter shell
Low resolution limit [Å]50.0003.010
High resolution limit [Å]2.9602.960
Rmerge0.0750.714
Number of reflections140161077
<I/σ(I)>18.71.1
Completeness [%]94.371.1
Redundancy4.94.2
Crystallization Conditions
crystal IDmethodpHtemperaturedetails
1VAPOR DIFFUSION, SITTING DROP72892% TACSIMATE, PH 7.0, 6% PEG3350

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