2YIX
Triazolopyridine Inhibitors of p38
Experimental procedure
Experimental method | SINGLE WAVELENGTH |
Source type | ROTATING ANODE |
Temperature [K] | 100 |
Spacegroup name | P 21 21 21 |
Unit cell lengths | 45.944, 86.523, 122.580 |
Unit cell angles | 90.00, 90.00, 90.00 |
Refinement procedure
Resolution | 24.750 - 2.300 |
R-factor | 0.1959 |
Rwork | 0.193 |
R-free | 0.24720 |
Structure solution method | OTHER |
Starting model (for MR) | NONE |
RMSD bond length | 0.010 |
RMSD bond angle | 1.130 |
Refinement software | BUSTER (2.9.6) |
Data quality characteristics
Overall | |
Low resolution limit [Å] | 25.000 |
High resolution limit [Å] | 2.300 |
Rmerge | 0.080 |
Number of reflections | 21609 |
<I/σ(I)> | 12 |
Completeness [%] | 96.0 |
Redundancy | 2.8 |
Crystallization Conditions
crystal ID | method | pH | temperature | details |
1 |