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2WI3

Orally Active 2-Amino Thienopyrimidine Inhibitors of the Hsp90 Chaperone

Experimental procedure
実験手法SINGLE WAVELENGTH
Source typeROTATING ANODE
Source detailsRIGAKU RUH3R
Temperature [K]100
Detector technologyIMAGE PLATE
Collection date2002-09-10
DetectorRIGAKU RAXIS IV
Spacegroup nameI 2 2 2
格子定数 [Å]65.682, 89.172, 99.783
格子定数 [度]90.00, 90.00, 90.00
精密化法
残基65.940 - 1.900
R因子0.19992
Rwork0.198
R-free0.24248
Structure solution methodMOLECULAR REPLACEMENT
Starting model (for MR)1uy6
結合長の平均二乗偏差(RMSD) [Å]0.028
結合角の平均二乗偏差(RMSD) [度]2.215
Data reduction softwared*TREK
Phasing softwareAMoRE
Refinement softwareREFMAC (5.5.0066)
Quality characteristics
 OverallOuter shell
分解能 [Å] (低)30.0002.250
分解能 [Å] (高)1.9001.900
Rmerge_l_obs0.0200.180
独立反射数21769
<I/σ(I)>21.23.2
完全性 [%]92.864
冗長性2
結晶化条件
結晶ID方法pH温度溶液条件
16.5pH 6.5

225158

件を2024-09-18に公開中

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