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1WS6
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BU of 1ws6 by Molmil
The Structure of Thermus thermphillus HB8 hypothetical protein TTHA0928
Descriptor: methyltransferase
Authors:Sasaki, C, Sugiura, I, Sugio, S, Tamura, T, Inagaki, K, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
Deposit date:2004-11-01
Release date:2006-02-07
Last modified:2024-10-30
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:The structure of thermus thermphillus HB8 hypothetical protein TTHA0928
TO BE PUBLISHED
2E1M
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BU of 2e1m by Molmil
Crystal Structure of L-Glutamate Oxidase from Streptomyces sp. X-119-6
Descriptor: FLAVIN-ADENINE DINUCLEOTIDE, L-glutamate oxidase, PHOSPHATE ION
Authors:Sasaki, C, Kashima, A, Sakaguchi, C, Mizuno, H, Arima, J, Kusakabe, H, Tamura, T, Sugio, S, Inagaki, K.
Deposit date:2006-10-26
Release date:2007-11-13
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Structural characterization of l-glutamate oxidase from Streptomyces sp. X-119-6
Febs J., 276, 2009
8YMI
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BU of 8ymi by Molmil
BRD4-BD1 in complex with 2-{[(3S)-1-benzylpyrrolidin-3-yl]methyl}-5-methyl-7-(1-methylpyrazol-3-yl)pyrazolo[4,3-c]pyridin-4-one
Descriptor: 1,2-ETHANEDIOL, 2-{[(3S)-1-benzylpyrrolidin-3-yl]methyl}-5-methyl-7-(1-methylpyrazol-3-yl)pyrazolo[4,3-c]pyridin-4-one, Bromodomain-containing protein 4
Authors:Sasaki, C, Miyaguchi, I, Hagihara, S, Ishizawa, K, Endo, J.
Deposit date:2024-03-09
Release date:2025-03-12
Method:X-RAY DIFFRACTION (1.01 Å)
Cite:Discovery of a potent, orally available pyrazolopyridone derivative as a novel selective BET BD1 Inhibitor (Part 2).
To Be Published
8YMG
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BU of 8ymg by Molmil
BRD4-BD1 in complex with 7-[4-chloro-1-(tetrahydropyran-4-ylmethyl)imidazol-2-yl]-5-methyl-2-{[(2R)-2-methyl-4-methylsulfonyl-piperazin-1-yl]methyl}furo[3,2-c]pyridin-4-one
Descriptor: 7-[4-chloro-1-(tetrahydropyran-4-ylmethyl)imidazol-2-yl]-5-methyl-2-{[(2R)-2-methyl-4-methylsulfonyl-piperazin-1-yl]methyl}furo[3,2-c]pyridin-4-one, Bromodomain-containing protein 4
Authors:Sasaki, C, Miyaguchi, I, Hagihara, S, Ishizawa, K, Endo, J.
Deposit date:2024-03-09
Release date:2025-03-12
Method:X-RAY DIFFRACTION (1.007 Å)
Cite:Discovery of a potent, orally available furopyridine derivative as a novel selective BET BD1 Inhibitor (Part 1).
To Be Published
8YMF
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BU of 8ymf by Molmil
BRD4-BD1 in complex with 7-[2-(cyclopropylmethoxy)phenyl]-5-methyl-2-[(1-methylsulfonyl-4-piperidyl)methyl]pyrazolo[4,3-c]pyridin-4-one
Descriptor: 7-[2-(cyclopropylmethoxy)phenyl]-5-methyl-2-[(1-methylsulfonylpiperidin-4-yl)methyl]pyrazolo[4,3-c]pyridin-4-one, Bromodomain-containing protein 4
Authors:Sasaki, C, Miyaguchi, I, Hagihara, S, Ishizawa, K, Endo, J.
Deposit date:2024-03-09
Release date:2025-03-12
Method:X-RAY DIFFRACTION (1.015 Å)
Cite:Discovery of a potent, orally available pyrazolopyridone derivative as a novel selective BET BD1 Inhibitor (Part 2).
To Be Published
8YMH
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BU of 8ymh by Molmil
BRD4-BD1 in complex with 5-methyl-2-{[(2R)-2-methyl-4-methylsulfonyl-piperazin-1-yl]methyl}-7-(1-methylpyrazol-3-yl)furo[3,2-c]pyridin-4-one
Descriptor: 1,2-ETHANEDIOL, 5-methyl-2-{[(2R)-2-methyl-4-methylsulfonyl-piperazin-1-yl]methyl}-7-(1-methylpyrazol-3-yl)furo[3,2-c]pyridin-4-one, Bromodomain-containing protein 4
Authors:Sasaki, C, Miyaguchi, I, Hagihara, S, Ishizawa, K, Endo, J.
Deposit date:2024-03-09
Release date:2025-03-12
Method:X-RAY DIFFRACTION (1.04 Å)
Cite:Discovery of a potent, orally available furopyridine derivative as a novel selective BET BD1 Inhibitor (Part 1).
To Be Published
8YME
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BU of 8yme by Molmil
BRD4-BD1 in complex with N-cyclohexyl-1-methyl-6-{[5-methyl-7-(1-methylpyrazol-3-yl)-4-oxo-pyrazolo[4,3-c]pyridin-2-yl]methyl}azepan-1-ium-4-carboxamide 2,2,2-trifluoroacetate
Descriptor: (4R,6S)-N-cyclohexyl-1-methyl-6-[[5-methyl-7-(1-methylpyrazol-3-yl)-4-oxidanylidene-pyrazolo[4,3-c]pyridin-2-yl]methyl]azepane-4-carboxamide, 1,2-ETHANEDIOL, Bromodomain-containing protein 4, ...
Authors:Sasaki, C, Miyaguchi, I, Hagihara, S, Ishizawa, K, Endo, J.
Deposit date:2024-03-09
Release date:2025-03-12
Method:X-RAY DIFFRACTION (1.18 Å)
Cite:Discovery of a potent, orally available pyrazolopyridone derivative as a novel selective BET BD1 Inhibitor (Part 2).
To Be Published
1RTU
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BU of 1rtu by Molmil
USTILAGO SPHAEROGENA RIBONUCLEASE U2
Descriptor: RIBONUCLEASE U2, SULFATE ION
Authors:Noguchi, S, Satow, Y, Uchida, T, Sasaki, C, Matsuzaki, T.
Deposit date:1995-05-12
Release date:1996-11-08
Last modified:2024-11-13
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Crystal structure of Ustilago sphaerogena ribonuclease U2 at 1.8 A resolution.
Biochemistry, 34, 1995
1J1C
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BU of 1j1c by Molmil
Binary complex structure of human tau protein kinase I with ADP
Descriptor: ADENOSINE-5'-DIPHOSPHATE, Glycogen synthase kinase-3 beta, MAGNESIUM ION
Authors:Aoki, M, Yokota, T, Sugiura, I, Sasaki, C, Hasegawa, T, Okumura, C, Kohno, T, Sugio, S, Matsuzaki, T.
Deposit date:2002-12-03
Release date:2003-12-03
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Structural insight into nucleotide recognition in tau-protein kinase I/glycogen synthase kinase 3 beta.
Acta Crystallogr.,Sect.D, 60, 2004
1J1B
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BU of 1j1b by Molmil
Binary complex structure of human tau protein kinase I with AMPPNP
Descriptor: Glycogen synthase kinase-3 beta, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
Authors:Aoki, M, Yokota, T, Sugiura, I, Sasaki, C, Hasegawa, T, Okumura, C, Kohno, T, Sugio, S, Matsuzaki, T.
Deposit date:2002-12-03
Release date:2003-12-03
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Structural insight into nucleotide recognition in tau-protein kinase I/glycogen synthase kinase 3 beta.
Acta Crystallogr.,Sect.D, 60, 2004
2DY3
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BU of 2dy3 by Molmil
Crystal Structure of alanine racemase from Corynebacterium glutamicum
Descriptor: Alanine racemase, PYRIDOXAL-5'-PHOSPHATE
Authors:Miyaguchi, I, Sasaki, C, Kato, R, Oikawa, T, Sugio, S.
Deposit date:2006-09-05
Release date:2007-09-11
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Crystal Structure of Alanine Racemase from Corynebacterium glutamicum at 2.1 A resolution
To be Published
1J1J
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BU of 1j1j by Molmil
Crystal Structure of human Translin
Descriptor: Translin
Authors:Sugiura, I, Sasaki, C, Hasegawa, T, Kohno, T, Sugio, S, Moriyama, H, Kasai, M, Matsuzaki, T.
Deposit date:2002-12-06
Release date:2003-12-06
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Structure of human translin at 2.2 A resolution.
Acta Crystallogr.,Sect.D, 60, 2004

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