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1ZTZ
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BU of 1ztz by Molmil
Crystal structure of HIV protease- metallacarborane complex
Descriptor: COBALT BIS(1,2-DICARBOLLIDE), PROTEASE RETROPEPSIN, autoproteolytic tetrapeptide
Authors:Cigler, P, Kozisek, M, Rezacova, P, Brynda, J, Otwinowski, Z, Sedlacek, J, Bodem, J, Kraeusslich, H.-G, Kral, V, Konvalinka, J.
Deposit date:2005-05-28
Release date:2005-11-01
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:From nonpeptide toward noncarbon protease inhibitors: Metallacarboranes as specific and potent inhibitors of HIV protease
Proc.Natl.Acad.Sci.USA, 102, 2005
3T3C
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BU of 3t3c by Molmil
Structure of HIV PR resistant patient derived mutant (comprising 22 mutations) in complex with DRV
Descriptor: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, BETA-MERCAPTOETHANOL, HIV-1 protease, ...
Authors:Rezacova, P, Kozisek, M, Konvalinka, J, Saskova, K.G.
Deposit date:2011-07-25
Release date:2012-06-20
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Mutations in HIV-1 gag and pol Compensate for the Loss of Viral Fitness Caused by a Highly Mutated Protease.
Antimicrob.Agents Chemother., 56, 2012
2BUO
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BU of 2buo by Molmil
HIV-1 capsid C-terminal domain in complex with an inhibitor of particle assembly
Descriptor: ACETIC ACID, HIV-1 CAPSID PROTEIN, INHIBITOR OF CAPSID ASSEMBLY
Authors:Ternois, F, Sticht, J, Duquerroy, S, Krausslich, H.-G, Rey, F.A.
Deposit date:2005-06-17
Release date:2005-07-21
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:The HIV-1 Capsid Protein C-Terminal Domain in Complex with a Virus Assembly Inhibitor
Nat.Struct.Mol.Biol., 12, 2005

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