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4PM0
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BU of 4pm0 by Molmil
PDE7A catalytic domain in complex with 2-(Cyclopentylamino)thieno[3,2-d]pyrimidin-4(3H)-one derivative
Descriptor: 2-(cyclopentylamino)-3-ethyl-7-ethynylthieno[3,2-d]pyrimidin-4(3H)-one, High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A, MAGNESIUM ION, ...
Authors:Kawai, K, Endo, Y, Asano, T, Amano, S, Sawada, K, Ueo, N, Takahashi, N, Sonoda, Y, Kamei, N, Nagata, N.
Deposit date:2014-05-20
Release date:2014-12-03
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Discovery of 2-(Cyclopentylamino)thieno[3,2-d]pyrimidin-4(3H)-one Derivatives as a New Series of Potent Phosphodiesterase 7 Inhibitors.
J.Med.Chem., 57, 2014
7E5O
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BU of 7e5o by Molmil
Crystal structure of SARS-CoV-2 RBD in complex with antibody NT-193
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, NT-193 Heavy chain, NT-193 Light chain, ...
Authors:Kita, S, Onodera, T, Adachi, Y, Moriayma, S, Nomura, T, Tadokoro, T, Anraku, Y, Yumoto, K, Tian, C, Fukuhara, H, Suzuki, T, Tonouchi, K, Sasaki, J, Sun, L, Hashiguchi, T, Takahashi, Y, Maenaka, K.
Deposit date:2021-02-19
Release date:2021-09-08
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:A SARS-CoV-2 antibody broadly neutralizes SARS-related coronaviruses and variants by coordinated recognition of a virus-vulnerable site.
Immunity, 54, 2021
3WIL
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BU of 3wil by Molmil
Crystal structure of the CK2alpha/compound3 complex
Descriptor: Casein kinase II subunit alpha, {[(2Z)-2-(3,4-dimethoxybenzylidene)-3-oxo-2,3-dihydro-1-benzofuran-6-yl]oxy}acetic acid
Authors:Kinoshita, T, Nakanishi, I.
Deposit date:2013-09-18
Release date:2014-09-24
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:Identification of protein kinase CK2 inhibitors using solvent dipole ordering virtual screening
To be Published
3WIK
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BU of 3wik by Molmil
Crystal structure of the CK2alpha/compound10 complex
Descriptor: Casein kinase II subunit alpha, N-[5-(4-nitrophenyl)-1,3,4-thiadiazol-2-yl]acetamide
Authors:Kinoshita, T, Nakaniwa, T, Sekiguchi, Y, Nakanishi, I.
Deposit date:2013-09-18
Release date:2014-11-05
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (1.995 Å)
Cite:Identification of protein kinase CK2 inhibitors using solvent dipole ordering virtual screening
To be Published

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PDB entries from 2024-09-18

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