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5ZNI
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BU of 5zni by Molmil
Plasmodium falciparum purine nucleoside phosphorylase in complex with mefloquine
Descriptor: Mefloquine, PHOSPHATE ION, Purine nucleoside phosphorylase
Authors:Chen, D, Nordlund, P, Dziekan, J.M.
Deposit date:2018-04-09
Release date:2019-01-16
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Identifying purine nucleoside phosphorylase as the target of quinine using cellular thermal shift assay.
Sci Transl Med, 11, 2019
5ZNC
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BU of 5znc by Molmil
Plasmodium falciparum purine nucleoside phosphorylase in complex with quinine
Descriptor: PHOSPHATE ION, Purine nucleoside phosphorylase, Quinine
Authors:Chen, D, Nordlund, P.
Deposit date:2018-04-08
Release date:2019-01-16
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (1.66 Å)
Cite:Identifying purine nucleoside phosphorylase as the target of quinine using cellular thermal shift assay.
Sci Transl Med, 11, 2019
8HO4
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BU of 8ho4 by Molmil
Falcilysin in complex with MMV000848
Descriptor: (2R)-1-(9H-carbazol-9-yl)-3-(cyclopentylamino)propan-2-ol, 1,2-ETHANEDIOL, Falcilysin, ...
Authors:Lin, J.Q, Chung, Z, Lescar, J.
Deposit date:2022-12-09
Release date:2023-12-20
Last modified:2024-07-03
Method:X-RAY DIFFRACTION (1.96 Å)
Cite:Identification of an inhibitory pocket in falcilysin provides a new avenue for malaria drug development.
Cell Chem Biol, 31, 2024
8HO5
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BU of 8ho5 by Molmil
Falcilysin in complex with MMV665806
Descriptor: (2S)-1-(2,3-dimethyl-1H-indol-1-yl)-3-{[(1S,2S)-2-methylcyclohexyl]amino}propan-2-ol, 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, ...
Authors:Lin, J.Q, Chung, Z, Lescar, J.
Deposit date:2022-12-09
Release date:2023-12-20
Last modified:2024-07-03
Method:X-RAY DIFFRACTION (2.003 Å)
Cite:Identification of an inhibitory pocket in falcilysin provides a new avenue for malaria drug development.
Cell Chem Biol, 31, 2024
7DIJ
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BU of 7dij by Molmil
Falcilysin in complex with MK-4815
Descriptor: 1,2-ETHANEDIOL, 2-(aminomethyl)-3,5-ditert-butyl-phenol, ACETATE ION, ...
Authors:Lin, J.Q, El Sahili, A, Lescar, J.
Deposit date:2020-11-19
Release date:2021-12-01
Last modified:2024-05-29
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Identification of an inhibitory pocket in falcilysin provides a new avenue for malaria drug development.
Cell Chem Biol, 31, 2024
7DIA
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BU of 7dia by Molmil
Falcilysin in complex with mefloquine
Descriptor: (S)-[2,8-bis(trifluoromethyl)quinolin-4-yl]-[(2S)-piperidin-2-yl]methanol, 1,2-ETHANEDIOL, ACETATE ION, ...
Authors:Lin, J.Q, El Sahili, A, Lescar, J.
Deposit date:2020-11-18
Release date:2021-12-01
Last modified:2024-05-29
Method:X-RAY DIFFRACTION (1.55 Å)
Cite:Identification of an inhibitory pocket in falcilysin provides a new avenue for malaria drug development.
Cell Chem Biol, 31, 2024
7DI7
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BU of 7di7 by Molmil
Falcilysin in complex with chloroquine
Descriptor: ACETATE ION, Falcilysin, N4-(7-CHLORO-QUINOLIN-4-YL)-N1,N1-DIETHYL-PENTANE-1,4-DIAMINE, ...
Authors:Lin, J.Q, El Sahili, A, Lescar, J.
Deposit date:2020-11-18
Release date:2021-12-01
Last modified:2024-05-29
Method:X-RAY DIFFRACTION (1.82 Å)
Cite:Identification of an inhibitory pocket in falcilysin provides a new avenue for malaria drug development.
Cell Chem Biol, 31, 2024
8W7H
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BU of 8w7h by Molmil
Purine Nucleoside Phosphorylase in complex with MMV000848
Descriptor: (2R)-1-(9H-carbazol-9-yl)-3-(cyclopentylamino)propan-2-ol, 1,2-ETHANEDIOL, PHOSPHATE ION, ...
Authors:Chung, Z, Lin, J.Q, Lescar, J.
Deposit date:2023-08-30
Release date:2024-01-17
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Identification and structural validation of purine nucleoside phosphorylase from Plasmodium falciparum as a target of MMV000848.
J.Biol.Chem., 300, 2023

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PDB entries from 2024-09-18

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