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5FKW
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BU of 5fkw by Molmil
cryo-EM structure of the E. coli replicative DNA polymerase complex bound to DNA (DNA polymerase III alpha, beta, epsilon)
分子名称: DNA POLYMERASE III ALPHA, DNA POLYMERASE III BETA, DNA POLYMERASE III EPSILON, ...
著者Fernandez-Leiro, R, Conrad, J, Scheres, S.H.W, Lamers, M.H.
登録日2015-10-20
公開日2015-11-25
最終更新日2019-02-27
実験手法ELECTRON MICROSCOPY (7.3 Å)
主引用文献cryo-EM structures of theE. colireplicative DNA polymerase reveal its dynamic interactions with the DNA sliding clamp, exonuclease andtau.
Elife, 4, 2015
5FXT
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BU of 5fxt by Molmil
Crystal Structure of Helicobacter pylori beta clamp in complex with Carprofen
分子名称: (2S)-2-(6-chloro-9H-carbazol-2-yl)propanoic acid, DNA POLYMERASE III SUBUNIT BETA
著者Pandey, P, Gourinath, S.
登録日2016-03-02
公開日2017-08-16
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献Screening of E. coli beta-clamp Inhibitors Revealed that Few Inhibit Helicobacter pylori More Effectively: Structural and Functional Characterization.
Antibiotics (Basel), 7, 2018
5FKV
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BU of 5fkv by Molmil
cryo-EM structure of the E. coli replicative DNA polymerase complex bound to DNA (DNA polymerase III alpha, beta, epsilon, tau complex)
分子名称: DNA POLYMERASE III BETA, DNA POLYMERASE III EPSILON, DNA POLYMERASE III SUBUNIT ALPHA, ...
著者Fernandez-Leiro, R, Conrad, J, Scheres, S.H.W, Lamers, M.H.
登録日2015-10-20
公開日2015-11-25
最終更新日2019-02-27
実験手法ELECTRON MICROSCOPY (8 Å)
主引用文献cryo-EM structures of theE. colireplicative DNA polymerase reveal its dynamic interactions with the DNA sliding clamp, exonuclease andtau.
Elife, 4, 2015
8DKD
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BU of 8dkd by Molmil
Sliding clamp from M. thermoresistibile
分子名称: Beta sliding clamp
著者Kapur, M.K, Gray, O.J, Honzatko, R.H, Nelson, S.N.
登録日2022-07-05
公開日2023-01-18
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Interaction of sliding clamp with mycobacterial polymerases
To Be Published
5FVE
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BU of 5fve by Molmil
Crystal Structure of Helicobacter pylori beta clamp in complex with 3, 4-Difluorobenzamide
分子名称: 3,4-difluorobenzamide, DNA POLYMERASE III SUBUNIT BETA
著者Pandey, P, Gourinath, S.
登録日2016-02-05
公開日2017-02-22
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献Screening of E. coli beta-clamp Inhibitors Revealed that Few Inhibit Helicobacter pylori More Effectively: Structural and Functional Characterization.
Antibiotics (Basel), 7, 2018
8DK9
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BU of 8dk9 by Molmil
Sliding-clamp-DinX peptide
分子名称: ACETYL GROUP, AMINO GROUP, Beta sliding clamp, ...
著者Kapur, M.K, Gray, O.J, Honzatko, R.H, Nelson, S.N.
登録日2022-07-05
公開日2023-01-18
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Interaction of sliding clamp with mycobacterial polymerases
To Be Published
8DJQ
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BU of 8djq by Molmil
Sliding-clamp-DnaE1 peptide
分子名称: ACETYL GROUP, AMINO GROUP, Beta sliding clamp, ...
著者Kapur, M.K, Gray, O.J, Honzatko, R.H, Nelson, S.N.
登録日2022-07-01
公開日2023-01-18
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Interaction of the sliding clamp with mycobacterial polymerases
To Be Published
5G4Q
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BU of 5g4q by Molmil
H.pylori Beta clamp in complex with 5-chloroisatin
分子名称: 5-chloro-1H-indole-2,3-dione, DNA POLYMERASE III SUBUNIT BETA
著者Pandey, P, Gourinath, S.
登録日2016-05-16
公開日2017-06-21
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Screening of E. coli beta-clamp Inhibitors Revealed that Few Inhibit Helicobacter pylori More Effectively: Structural and Functional Characterization.
Antibiotics (Basel), 7, 2018
5G48
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BU of 5g48 by Molmil
H.pylori Beta clamp in complex with Diflunisal
分子名称: 5-(2,4-DIFLUOROPHENYL)-2-HYDROXY-BENZOIC ACID, DNA POLYMERASE III SUBUNIT BETA
著者Pandey, P, Gourinath, S.
登録日2016-05-06
公開日2017-06-21
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.28 Å)
主引用文献Targeting the beta-clamp in Helicobacter pylori with FDA-approved drugs reveals micromolar inhibition by diflunisal.
FEBS Lett., 591, 2017
8DJ6
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BU of 8dj6 by Molmil
Sliding-clamp-ImuB peptide
分子名称: ACETATE ION, Beta sliding clamp, FORMIC ACID, ...
著者Kapur, M.K, Gray, O.J, Honzatko, R.H, Nelson, S.N.
登録日2022-06-30
公開日2023-07-26
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Interaction of sliding clamp with mycobacterial polymerases
To Be Published
4K3Q
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BU of 4k3q by Molmil
E. coli sliding clamp in complex with AcQLDAF
分子名称: (ACE)QLDAF, CALCIUM ION, DI(HYDROXYETHYL)ETHER, ...
著者Yin, Z, Oakley, A.J.
登録日2013-04-11
公開日2013-05-01
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K74
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BU of 4k74 by Molmil
The UmuC subunit of the E. coli DNA polymerase V shows a unique interaction with the beta-clamp processivity factor.
分子名称: DNA polymerase III subunit beta, UmuC peptide
著者Patoli, A.A, Winter, J.A, Bunting, K.A.
登録日2013-04-16
公開日2013-07-17
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The UmuC subunit of the E. coli DNA polymerase V shows a unique interaction with the beta-clamp processivity factor.
Bmc Struct.Biol., 13, 2013
4K3M
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BU of 4k3m by Molmil
E.coli sliding clamp in complex with AcALDLF peptide
分子名称: ALDLF, CALCIUM ION, DI(HYDROXYETHYL)ETHER, ...
著者Yin, Z, Oakley, A.J.
登録日2013-04-11
公開日2013-05-01
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K3O
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BU of 4k3o by Molmil
E. coli sliding clamp in complex with AcQADLF
分子名称: (ACE)QADLF, 1,2-ETHANEDIOL, CALCIUM ION, ...
著者Yin, Z, Oakley, A.J.
登録日2013-04-11
公開日2013-05-01
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K3K
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BU of 4k3k by Molmil
E. Coli sliding clamp in complex with (S)-2-(4-methylpentanamido)-3-phenylpropanoic acid
分子名称: CALCIUM ION, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ...
著者Yin, Z, Oakley, A.J.
登録日2013-04-10
公開日2013-05-01
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K3P
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BU of 4k3p by Molmil
E. coli sliding clamp in complex with AcQLALF
分子名称: (ACE)QLALF, 1,2-ETHANEDIOL, CALCIUM ION, ...
著者Yin, Z, Oakley, A.J.
登録日2013-04-11
公開日2013-05-01
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K3R
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BU of 4k3r by Molmil
E. coli sliding clamp in complex with AcQLDLA
分子名称: (ACE)QLDLA, CALCIUM ION, CHLORIDE ION, ...
著者Yin, Z, Oakley, A.J.
登録日2013-04-11
公開日2013-05-01
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K3L
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BU of 4k3l by Molmil
E. coli sliding clamp in complex with AcLF dipeptide
分子名称: 1,2-ETHANEDIOL, ACETYL GROUP, CALCIUM ION, ...
著者Yin, Z, Oakley, A.J.
登録日2013-04-10
公開日2013-05-01
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K3S
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BU of 4k3s by Molmil
E. coli sliding clamp in P1 crystal space group
分子名称: CALCIUM ION, DNA polymerase III subunit beta, O-ACETALDEHYDYL-HEXAETHYLENE GLYCOL, ...
著者Yin, Z, Oakley, A.J.
登録日2013-04-11
公開日2013-05-01
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4MJR
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BU of 4mjr by Molmil
E. coli sliding clamp in complex with (S)-Carprofen
分子名称: (2S)-2-(6-chloro-9H-carbazol-2-yl)propanoic acid, CALCIUM ION, CHLORIDE ION, ...
著者Yin, Z, Oakley, A.J.
登録日2013-09-04
公開日2013-09-18
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.62 Å)
主引用文献DNA replication is the target for the antibacterial effects of nonsteroidal anti-inflammatory drugs.
Chem.Biol., 21, 2014
4MJP
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BU of 4mjp by Molmil
E. coli sliding clamp in complex with (R)-Vedaprofen
分子名称: (2R)-2-(4-cyclohexylnaphthalen-1-yl)propanoic acid, CALCIUM ION, CHLORIDE ION, ...
著者Yin, Z, Oakley, A.J.
登録日2013-09-04
公開日2013-09-18
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.855 Å)
主引用文献DNA replication is the target for the antibacterial effects of nonsteroidal anti-inflammatory drugs.
Chem.Biol., 21, 2014
4MJQ
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BU of 4mjq by Molmil
E. coli sliding clamp in complex with Bromfenac
分子名称: 1,2-ETHANEDIOL, CALCIUM ION, CHLORIDE ION, ...
著者Yin, Z, Oakley, A.J.
登録日2013-09-04
公開日2013-09-18
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.73 Å)
主引用文献DNA replication is the target for the antibacterial effects of nonsteroidal anti-inflammatory drugs.
Chem.Biol., 21, 2014
4N96
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BU of 4n96 by Molmil
E. coli sliding clamp in complex with 6-nitroindazole
分子名称: 6-NITROINDAZOLE, CALCIUM ION, CHLORIDE ION, ...
著者Yin, Z, Oakley, A.J.
登録日2013-10-19
公開日2013-11-06
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Discovery of lead compounds targeting the bacterial sliding clamp using a fragment-based approach.
J.Med.Chem., 57, 2014
4N95
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BU of 4n95 by Molmil
E. coli sliding clamp in complex with 5-chloroindoline-2,3-dione
分子名称: 5-chloro-1H-indole-2,3-dione, CALCIUM ION, CHLORIDE ION, ...
著者Yin, Z, Oakley, A.J.
登録日2013-10-19
公開日2013-11-06
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Discovery of lead compounds targeting the bacterial sliding clamp using a fragment-based approach.
J.Med.Chem., 57, 2014
4N94
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BU of 4n94 by Molmil
E. coli sliding clamp in complex with 3,4-difluorobenzamide
分子名称: 1,2-ETHANEDIOL, 3,4-difluorobenzamide, CALCIUM ION, ...
著者Yin, Z, Oakley, A.J.
登録日2013-10-19
公開日2013-11-06
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.73 Å)
主引用文献Discovery of lead compounds targeting the bacterial sliding clamp using a fragment-based approach.
J.Med.Chem., 57, 2014

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