1GG8
DESIGN OF INHIBITORS OF GLYCOGEN PHOSPHORYLASE: A STUDY OF ALPHA-AND BETA-C-GLUCOSIDES AND 1-THIO-BETA-D-GLUCOSE COMPOUNDS
1GG8 の概要
エントリーDOI | 10.2210/pdb1gg8/pdb |
分子名称 | PROTEIN (GLYCOGEN PHOSPHORYLASE), ALPHA-D-GLUCOPYRANOSYL-2-CARBOXYLIC ACID AMIDE, PYRIDOXAL-5'-PHOSPHATE, ... (5 entities in total) |
機能のキーワード | glycogen phosphorylase, inhibitor complex, catalytic site, design, transferase |
由来する生物種 | Oryctolagus cuniculus (rabbit) |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 98093.73 |
構造登録者 | Watson, K.A.,Mitchell, E.P.,Johnson, L.N.,Son, J.C.,Bichard, C.J.,Orchard, M.G.,Fleet, G.W.,Oikonomakos, N.G.,Leonidas, D.D.,Kontou, M.,Papageorgiou, A.C. (登録日: 2000-07-30, 公開日: 2000-08-23, 最終更新日: 2023-08-09) |
主引用文献 | Watson, K.A.,Mitchell, E.P.,Johnson, L.N.,Son, J.C.,Bichard, C.J.,Orchard, M.G.,Fleet, G.W.,Oikonomakos, N.G.,Leonidas, D.D.,Kontou, M.,Papageorgioui, A. Design of inhibitors of glycogen phosphorylase: a study of alpha- and beta-C-glucosides and 1-thio-beta-D-glucose compounds. Biochemistry, 33:5745-5758, 1994 Cited by PubMed: 8180201DOI: 10.1021/bi00185a011 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.31 Å) |
構造検証レポート
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