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1QLQ
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BU of 1qlq by Molmil
Bovine Pancreatic Trypsin Inhibitor (BPTI) Mutant with Altered Binding Loop Sequence
分子名称: PANCREATIC TRYPSIN INHIBITOR, SULFATE ION
著者Czapinska, H, Krzywda, S, Sheldrick, G.M, Otlewski, J, Jaskolski, M.
登録日1999-09-10
公開日1999-10-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献High Resolution Structure of Bovine Pancreatic Trypsin Inhibitor with Altered Binding Loop Sequence
J.Mol.Biol., 295, 1999
6F1F
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BU of 6f1f by Molmil
The methylene thioacetal BPTI (Bovine Pancreatic Trypsin Inhibitor) mutant structure
分子名称: GLYCEROL, Pancreatic trypsin inhibitor, SULFATE ION
著者Lansky, S, Mousa, R, Metanis, N, Shoham, G.
登録日2017-11-21
公開日2018-07-18
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.716 Å)
主引用文献BPTI folding revisited: switching a disulfide into methylene thioacetal reveals a previously hidden path.
Chem Sci, 9, 2018
6YHY
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BU of 6yhy by Molmil
A lid blocking mechanism of a cone snail toxin revealed at the atomic level
分子名称: Conk-S1
著者Saikia, C, Altman-Gueta, H, Dym, O, Frolow, F, Gurevitz, M, Gordon, D, Reuveny, E, Karbat, I.
登録日2020-03-31
公開日2021-04-14
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献A Molecular Lid Mechanism of K + Channel Blocker Action Revealed by a Cone Peptide.
J.Mol.Biol., 433, 2021
6NAN
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BU of 6nan by Molmil
NMR structure determination of Ixolaris and Factor X interaction reveals a noncanonical mechanism of Kunitz inhibition
分子名称: Ixolaris
著者De Paula, V.S, Sgourakis, N.G, Francischetti, I.M.B, Almeida, F.C.L, Monteiro, R.Q, Valente, A.P.
登録日2018-12-06
公開日2019-06-12
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献NMR structure determination of Ixolaris and factor X(a) interaction reveals a noncanonical mechanism of Kunitz inhibition.
Blood, 134, 2019
6KZF
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BU of 6kzf by Molmil
Racemic X-ray Structure of Calcicludine
分子名称: D-calcicludine, Kunitz-type serine protease inhibitor homolog calcicludine
著者Qu, Q, Gao, S, Liu, L.
登録日2019-09-24
公開日2019-11-06
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.52 Å)
主引用文献Synthesis of Disulfide Surrogate Peptides Incorporating Large-Span Surrogate Bridges Through a Native-Chemical-Ligation-Assisted Diaminodiacid Strategy
Angew.Chem.Int.Ed.Engl., 59, 2020
5PTI
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BU of 5pti by Molmil
STRUCTURE OF BOVINE PANCREATIC TRYPSIN INHIBITOR. RESULTS OF JOINT NEUTRON AND X-RAY REFINEMENT OF CRYSTAL FORM II
分子名称: PHOSPHATE ION, TRYPSIN INHIBITOR, UNKNOWN ATOM OR ION
著者Wlodawer, A, Huber, R.
登録日1984-10-05
公開日1984-10-29
最終更新日2018-10-24
実験手法NEUTRON DIFFRACTION (1 Å), X-RAY DIFFRACTION
主引用文献Structure of bovine pancreatic trypsin inhibitor. Results of joint neutron and X-ray refinement of crystal form II
J.Mol.Biol., 180, 1984
2KNT
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BU of 2knt by Molmil
THE 1.2 ANGSTROM STRUCTURE OF KUNITZ TYPE DOMAIN C5
分子名称: COLLAGEN, PHOSPHATE ION
著者Merigeau, K, Arnoux, B, Ducruix, A.
登録日1997-01-15
公開日1997-05-15
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献1.2 A refinement of the Kunitz-type domain from the alpha3 chain of human type VI collagen.
Acta Crystallogr.,Sect.D, 54, 1998
4DTG
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BU of 4dtg by Molmil
Hemostatic effect of a monoclonal antibody mAb 2021 blocking the interaction between FXa and TFPI in a rabbit hemophilia model
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GLYCEROL, Humanized recombinant FAB fragment, ...
著者Svensson, L.A, Breinholt, J, Krogh, B.O, Hilden, I.
登録日2012-02-21
公開日2012-06-13
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Hemostatic effect of a monoclonal antibody mAb 2021 blocking the interaction between FXa and TFPI in a rabbit hemophilia model.
Blood, 119, 2012
9PTI
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BU of 9pti by Molmil
BASIC PANCREATIC TRYPSIN INHIBITOR (MET 52 OXIDIZED)
分子名称: BOVINE PANCREATIC TRYPSIN INHIBITOR, PHOSPHATE ION
著者Eigenbrot, C, Randal, M, Kossiakoff, A.A.
登録日1991-04-08
公開日1992-04-15
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (1.22 Å)
主引用文献

5XX2
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BU of 5xx2 by Molmil
A BPTI-[5,55] variant with C14GA38L mutations
分子名称: Pancreatic trypsin inhibitor, SULFATE ION
著者Islam, M.M.
登録日2017-07-01
公開日2018-07-04
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.12 Å)
主引用文献Hydrophobic surface residues can stabilize a protein through improved water-protein interactions.
Febs J., 2019
5XX4
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BU of 5xx4 by Molmil
A BPTI-[5,55] variant with C14GA38K mutations
分子名称: Pancreatic trypsin inhibitor, SULFATE ION
著者Islam, M.M.
登録日2017-07-01
公開日2018-07-04
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献Hydrophobic surface residues can stabilize a protein through improved water-protein interactions.
Febs J., 2019
5XX5
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BU of 5xx5 by Molmil
A BPTI-[5,55] variant with C14GA38I mutations
分子名称: Pancreatic trypsin inhibitor, SULFATE ION
著者Islam, M.M.
登録日2017-07-01
公開日2018-07-04
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.38 Å)
主引用文献Hydrophobic surface residues can stabilize a protein through improved water-protein interactions.
Febs J., 2019
5NMV
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BU of 5nmv by Molmil
Crystal structure of 2F22 Fab fragment against TFPI1
分子名称: Fab heavy chain, Fab light chain, GLYCEROL, ...
著者Svensson, L.A, Petersen, H.H.
登録日2017-04-07
公開日2018-03-28
最終更新日2018-05-09
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Factor Xa and VIIa inhibition by tissue factor pathway inhibitor is prevented by a monoclonal antibody to its Kunitz-1 domain.
J. Thromb. Haemost., 16, 2018
6PTI
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BU of 6pti by Molmil
STRUCTURE OF FORM III CRYSTALS OF BOVINE PANCREATIC TRYPSIN INHIBITOR
分子名称: PANCREATIC TRYPSIN INHIBITOR PRECURSOR, PHOSPHATE ION
著者Wlodawer, A.
登録日1987-05-13
公開日1987-10-16
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structure of form III crystals of bovine pancreatic trypsin inhibitor.
J.Mol.Biol., 198, 1987
6Q6C
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BU of 6q6c by Molmil
Pore-modulating toxins exploit inherent slow inactivation to block K+ channels
分子名称: 1,2-ETHANEDIOL, Kunitz-type conkunitzin-S1, NITRATE ION, ...
著者Karbat, I, Gueta, H, Fine, S, Szanto, T, Hamer-Rogotner, S, Dym, O, Frolow, F, Gordon, D, Panyi, G, Gurevitz, M, Reuveny, E.
登録日2018-12-10
公開日2019-08-21
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Pore-modulating toxins exploit inherent slow inactivation to block K+channels.
Proc.Natl.Acad.Sci.USA, 116, 2019
6Q61
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BU of 6q61 by Molmil
Pore-modulating toxins exploit inherent slow inactivation to block K+ channels
分子名称: Kunitz-type conkunitzin-S1, SULFATE ION
著者Karbat, I, Gueta, H, Fine, S, Szanto, T, Hamer-Rogotner, S, Dym, O, Frolow, F, Gordon, D, Panyi, G, Gurevitz, M, Reuveny, E.
登録日2018-12-10
公開日2019-08-21
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Pore-modulating toxins exploit inherent slow inactivation to block K+channels.
Proc.Natl.Acad.Sci.USA, 116, 2019
5JB6
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BU of 5jb6 by Molmil
A simplified BPTI variant containing 23 alanines out of 58 residues
分子名称: Pancreatic trypsin inhibitor, SULFATE ION
著者Islam, M.M.
登録日2016-04-13
公開日2017-04-19
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structures of highly simplified BPTIs provide insights into hydration-driven increase of unfolding enthalpy
Sci Rep, 7, 2017
5JB4
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BU of 5jb4 by Molmil
A simplified BPTI variant containing 21 alanines out 58 of residues
分子名称: Pancreatic trypsin inhibitor, SULFATE ION
著者Islam, M.M.
登録日2016-04-13
公開日2017-04-19
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Crystal structures of highly simplified BPTIs provide insights into hydration-driven increase of unfolding enthalpy
Sci Rep, 7, 2017
2DDI
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BU of 2ddi by Molmil
NMR structure of the second Kunitz domain of human WFIKKN1
分子名称: WAP, follistatin/kazal, immunoglobulin, ...
著者Liepinsh, E, Otting, G.
登録日2006-01-30
公開日2006-12-19
最終更新日2022-03-09
実験手法SOLUTION NMR
主引用文献Second Kunitz-type protease inhibitor domain of the human WFIKKN1 protein
J.Biomol.Nmr, 35, 2006
2M99
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BU of 2m99 by Molmil
Solution structure of a chymotrypsin inhibitor from the Taiwan cobra
分子名称: Protease inhibitor NACI
著者Lin, Y.-J, Ikeya, T, Guntert, P, Chang, L.-S.
登録日2013-06-05
公開日2013-10-16
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献NMR solution structure of a Chymotrypsin inhibitor from the Taiwan cobra Naja naja atra.
Molecules, 18, 2013
2DDJ
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BU of 2ddj by Molmil
NMR structure of the second Kunitz domain of human WFIKKN1
分子名称: WAP, follistatin/kazal, immunoglobulin, ...
著者Liepinsh, E, Otting, G.
登録日2006-01-30
公開日2006-12-19
最終更新日2022-03-09
実験手法SOLUTION NMR
主引用文献Second Kunitz-type protease inhibitor domain of the human WFIKKN1 protein
J.Biomol.Nmr, 35, 2006
2M01
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BU of 2m01 by Molmil
Solution structure of Kunitz-type neurotoxin LmKKT-1a from scorpion venom
分子名称: Protease inhibitor LmKTT-1a
著者Luo, F, Jiang, L, Liu, M, Chen, Z, Wu, Y.
登録日2012-10-15
公開日2013-11-13
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Genomic and structural characterization of Kunitz-type peptide LmKTT-1a highlights diversity and evolution of scorpion potassium channel toxins.
Plos One, 8, 2013
3OFW
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BU of 3ofw by Molmil
Crystal structure of recombinant Kunitz Type serine protease Inhibitor-1 from the Carribean sea anemone stichodactyla helianthus
分子名称: CHLORIDE ION, Kunitz-type proteinase inhibitor SHPI-1
著者Garcia-Fernandez, R, Redecke, L, Pons, T, Perbandt, M, Talavera, A, Gil, D, Gonzalez, Y, de los Angeles Chavez, M, Betzel, C.
登録日2010-08-16
公開日2011-08-17
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structure of the recombinant BPTI/Kunitz-type inhibitor rShPI-1A from the marine invertebrate Stichodactyla helianthus.
Acta Crystallogr.,Sect.F, 68, 2012
5JB7
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BU of 5jb7 by Molmil
A simplified BPTI variant containing 24 alanines out of 58 residues
分子名称: Pancreatic trypsin inhibitor, SULFATE ION
著者Islam, M.M.
登録日2016-04-13
公開日2017-04-19
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structures of highly simplified BPTIs provide insights into hydration-driven increase of unfolding enthalpy
Sci Rep, 7, 2017
5JB5
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BU of 5jb5 by Molmil
A simplified BPTI variant containing 22 alanines out of 58 residues
分子名称: Pancreatic trypsin inhibitor, SULFATE ION
著者Islam, M.M.
登録日2016-04-13
公開日2017-04-19
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Crystal structures of highly simplified BPTIs provide insights into hydration-driven increase of unfolding enthalpy
Sci Rep, 7, 2017

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