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6PKC

Inhibition of Human Menin by VTP-50469

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
B0005634cellular_componentnucleus
Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue OP4 A 601
ChainResidue
ASER155
ATYR319
AMET322
ATYR323
ATRP341
AGLU363
AVAL367
AHOH777
ASER178
AGLU179
AHIS181
AALA182
APHE238
ACYS241
ATYR276
AMET278

site_idAC2
Number of Residues19
Detailsbinding site for residue OP4 B 601
ChainResidue
BSER155
BSER178
BGLU179
BHIS181
BALA182
BPHE238
BCYS241
BTYR276
BMET278
BTYR319
BMET322
BTYR323
BTRP341
BVAL367
BHOH705
BHOH719
BHOH810
BHOH813
BHOH841

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:24275569
ChainResidueDetails
AALA581
BALA581

site_idSWS_FT_FI2
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails

219869

PDB entries from 2024-05-15

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