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5MWJ

Structure Enabled Discovery of a Stapled Peptide Inhibitor to Target the Oncogenic Transcriptional Repressor TLE1

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue DMS A 801
ChainResidue
ATHR496
AARG497
AILE512
ASER513
ATYR753

site_idAC2
Number of Residues14
Detailsbinding site for residue EBU A 802
ChainResidue
AGLU550
APRO575
AALA576
ATYR578
ASER620
ALEU636
APHE661
ALYS718
ALEU743
AHOH923
ACYS488
AASN531
ATYR532
AARG534

site_idAC3
Number of Residues7
Detailsbinding site for residue EBU B 801
ChainResidue
BCYS488
BARG534
BTYR578
BLEU636
BPHE661
BLEU702
BLEU743

Functional Information from PROSITE/UniProt
site_idPS00678
Number of Residues15
DetailsWD_REPEATS_1 Trp-Asp (WD) repeats signature. CFSCcsDgNIAVWDL
ChainResidueDetails
ACYS589-LEU603
ALEU631-LEU645

218853

PDB entries from 2024-04-24

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