PDB: 2569 resultsInfo pagesStatus searchChemie searchBIRD

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6XVD	Crystal structure of complex of urokinase and a upain-1 variant(W3F) in pH7.4 condition Descriptor: Urokinase-type plasminogen activator, upain-1-W3F Authors: Xue, G.P, Xie, X, Zhou, Y, Yuan, C, Huang, M.D, Jiang, L.G. Deposit date: 2020-01-21 Release date: 2020-02-19 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.4 Å) Cite: Insight to the residue in P2 position prevents the peptide inhibitor from being hydrolyzed by serine proteases. Biosci.Biotechnol.Biochem., 84, 2020
6XYK	Crystal structure of bovine trypsin at room temperature. Descriptor: BENZAMIDINE, CALCIUM ION, Cationic trypsin, ... Authors: Jensen, M. Deposit date: 2020-01-30 Release date: 2021-01-27 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.50000036 Å) Cite: Femtosecond structure of bovine trypsin at room temperature To Be Published
6XYG	Femtosecond structure of bovine trypsin at room temperature Descriptor: BENZAMIDINE, CALCIUM ION, Cationic trypsin, ... Authors: Jensen, M. Deposit date: 2020-01-30 Release date: 2021-02-10 Last modified: 2024-02-07 Method: X-RAY DIFFRACTION (1.50000238 Å) Cite: High-resolution macromolecular crystallography at the FemtoMAX beamline with time-over-threshold photon detection J.Synchrotron Radiat., 2021
6YIV	Trypsin inhibitor in complex with bovine trypsin Descriptor: Cationic trypsin, DIMETHYL SULFOXIDE, SULFATE ION, ... Authors: Badran, M.J, Heine, A, Klebe, G. Deposit date: 2020-04-01 Release date: 2020-12-02 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (0.95 Å) Cite: Trypsin inhibitor in complex with bovine trypsin To Be Published
6YIX	Trypsin inhibitor in complex with bovine trypsin Descriptor: Cationic trypsin, DIMETHYL SULFOXIDE, SULFATE ION, ... Authors: Badran, M.J, Heine, A, Klebe, G. Deposit date: 2020-04-01 Release date: 2020-12-02 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.31 Å) Cite: Trypsin inhibitor in complex with bovine trypsin To Be Published
6YIW	Trypsin inhibitor in complex with bovine trypsin Descriptor: 1H-isoindol-3-amine, CALCIUM ION, Cationic trypsin, ... Authors: Badran, M.J, Heine, A, Klebe, G. Deposit date: 2020-04-01 Release date: 2020-12-02 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (0.97 Å) Cite: Trypsin inhibitor in complex with bovine trypsin To Be Published
6Y4S	Human kallikrein-related peptidase 7 (KLK7) in the unliganded state Descriptor: Kallikrein-7, SULFATE ION, TRIETHYLENE GLYCOL Authors: Hanke, S, Strater, N. Deposit date: 2020-02-23 Release date: 2020-05-20 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (2.23 Å) Cite: Structural Studies on the Inhibitory Binding Mode of Aromatic Coumarinic Esters to Human Kallikrein-Related Peptidase 7. J.Med.Chem., 63, 2020
6YIS	Trypsin inhibitor in complex with bovine trypsin Descriptor: CALCIUM ION, Cationic Trypsin, DIMETHYL SULFOXIDE, ... Authors: Badran, M.J, Heine, A, Klebe, G. Deposit date: 2020-04-01 Release date: 2020-12-02 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.19 Å) Cite: Trypsin inhibitor in complex with bovine trypsin To Be Published
6YIT	Trypsin inhibitor in complex with bovine trypsin Descriptor: CALCIUM ION, Cationic trypsin, DIMETHYL SULFOXIDE, ... Authors: Badran, M.J, Heine, A, Klebe, G. Deposit date: 2020-04-01 Release date: 2020-12-02 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.25 Å) Cite: Trypsin inhibitor in complex with bovine trypsin To Be Published
6YIY	Trypsin inhibitor in complex with bovine trypsin Descriptor: 1H-isoindol-3-amine, CALCIUM ION, Cationic trypsin, ... Authors: Badran, M.J, Heine, A, Klebe, G. Deposit date: 2020-04-01 Release date: 2020-12-02 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.11 Å) Cite: Trypsin inhibitor in complex with bovine trypsin To Be Published
6YIU	Trypsin inhibitor in complex with bovine trypsin Descriptor: 3-aminobenzamide, CALCIUM ION, Cationic trypsin, ... Authors: Badran, M.J, Heine, A, Klebe, G. Deposit date: 2020-04-01 Release date: 2020-12-02 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.36 Å) Cite: Trypsin inhibitor in complex with bovine trypsin To Be Published
6YDY	Cationic Trypsin in Complex with a D-Phe-Pro-benzylamine derivative Descriptor: (2~{S})-~{N}-[[4-(aminomethyl)phenyl]methyl]-1-[(2~{R})-2-azanyl-3-phenyl-propanoyl]pyrrolidine-2-carboxamide, CALCIUM ION, Cationic Trypsin Authors: Ngo, K, Heine, A, Klebe, G. Deposit date: 2020-03-21 Release date: 2021-03-31 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.45 Å) Cite: Cationic Trypsin in Complex with a D-Phe-Pro-benzylamine derivative To Be Published
6YZC	Trypsin inhibitor in complex with bovine trypsin Descriptor: 1,2-ETHANEDIOL, CALCIUM ION, Cationic trypsin, ... Authors: Badran, M.J, Heine, A, Klebe, G. Deposit date: 2020-05-06 Release date: 2020-12-02 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.42 Å) Cite: Trypsin inhibitor in complex with bovine trypsin To Be Published
6ZFK	Trypsin inhibitor in complex with bovine trypsin Descriptor: 4-oxo-N-[(1S)-1-(pyridin-3-yl)ethyl]-4-(thiophen-2-yl)butanamide, CALCIUM ION, Cationic trypsin, ... Authors: Badran, M.J, Heine, A, Klebe, G. Deposit date: 2020-06-17 Release date: 2021-01-13 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.1 Å) Cite: Trypsin inhibitor in complex with bovine trypsin To Be Published
6ZFJ	Trypsin inhibitor in complex with bovine trypsin Descriptor: 1H-isoindol-3-amine, CALCIUM ION, Cationic trypsin, ... Authors: Badran, M.J, Heine, A, Klebe, G. Deposit date: 2020-06-17 Release date: 2021-01-13 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1 Å) Cite: Trypsin inhibitor in complex with bovine trypsin To Be Published
6YZA	Trypsin inhibitor in complex with bovine trypsin Descriptor: 1,2-ETHANEDIOL, CALCIUM ION, Cationic trypsin, ... Authors: Badran, M.J, Heine, A, Klebe, G. Deposit date: 2020-05-06 Release date: 2020-12-02 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.3 Å) Cite: Trypsin inhibitor in complex with bovine trypsin To Be Published
6CHA	STRUCTURE OF A TETRAHEDRAL TRANSITION STATE COMPLEX OF ALPHA-*CHYMOTRYPSIN AT 1.8-*ANGSTROMS RESOLUTION Descriptor: ALPHA-CHYMOTRYPSIN A, PHENYLETHANE BORONIC ACID Authors: Tulinsky, A, Blevins, R.A. Deposit date: 1987-02-06 Release date: 1987-04-16 Last modified: 2011-07-13 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Structure of a tetrahedral transition state complex of alpha-chymotrypsin dimer at 1.8-A resolution. J.Biol.Chem., 262, 1987
6D3Z	Protease SFTI complex Descriptor: Plasminogen, Trypsin inhibitor 1 Authors: Law, R.H.P, Wu, G. Deposit date: 2018-04-17 Release date: 2019-01-23 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (2 Å) Cite: Highly Potent and Selective Plasmin Inhibitors Based on the Sunflower Trypsin Inhibitor-1 Scaffold Attenuate Fibrinolysis in Plasma. J. Med. Chem., 62, 2019
6DI8	Crystal structure of bovine alpha-chymotrypsin in space group P65 Descriptor: Chymotrypsin A chain A, Chymotrypsin A chain B, Chymotrypsin A chain C, ... Authors: Marshall, A.C, Keiller, B.G, Bruning, J.B. Deposit date: 2018-05-23 Release date: 2019-01-23 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (1.859 Å) Cite: Crystal Structure of Bovine Alpha-Chymotrypsin in Space Group P65 Crystals, 8, 2018
6D40	Highly Potent and Selective Plasmin Inhibitors Based on the Sunflower Trypsin Inhibitor-1 Scaffold Attenuate Fibrinolysis in Plasma Descriptor: Plasminogen, SULFATE ION, Trypsin inhibitor 1 Authors: Law, R.H.P, Wu, G. Deposit date: 2018-04-17 Release date: 2019-01-23 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (1.43 Å) Cite: Highly Potent and Selective Plasmin Inhibitors Based on the Sunflower Trypsin Inhibitor-1 Scaffold Attenuate Fibrinolysis in Plasma. J. Med. Chem., 62, 2019
6D3Y	Highly Potent and Selective Plasmin Inhibitors Based on the Sunflower Trypsin Inhibitor-1 Scaffold Attenuate Fibrinolysis in Plasma Descriptor: GLYCEROL, Plasminogen, SULFATE ION, ... Authors: Law, R.H.P, Wu, G. Deposit date: 2018-04-17 Release date: 2019-01-23 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (1.32 Å) Cite: Highly Potent and Selective Plasmin Inhibitors Based on the Sunflower Trypsin Inhibitor-1 Scaffold Attenuate Fibrinolysis in Plasma. J. Med. Chem., 62, 2019
6D3X	Highly Potent and Selective Plasmin Inhibitors Based on the Sunflower Trypsin Inhibitor-1 Scaffold Attenuate Fibrinolysis in Plasma Descriptor: Plasminogen, Trypsin inhibitor 1 Authors: Law, R.H.P, Wu, G. Deposit date: 2018-04-17 Release date: 2019-01-23 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Highly Potent and Selective Plasmin Inhibitors Based on the Sunflower Trypsin Inhibitor-1 Scaffold Attenuate Fibrinolysis in Plasma. J. Med. Chem., 62, 2019
6DWR	Trypsin serine protease modified with the protease inhibitor cyanobenzylsulfonylfluoride Descriptor: 1,2-ETHANEDIOL, CALCIUM ION, Cationic trypsin, ... Authors: Luo, M, Eaton, C.N, Phillips-Piro, C.M. Deposit date: 2018-06-27 Release date: 2019-07-03 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (1.319 Å) Cite: Paired Spectroscopic and Crystallographic Studies of Protease Active Sites Chemistryselect, 4, 2019
6DZF	Orthorhombic trypsin cryocooled to 100 K with 20% xylose as cryoprotectant Descriptor: BENZAMIDINE, CALCIUM ION, Cationic trypsin, ... Authors: Juers, D.H. Deposit date: 2018-07-03 Release date: 2018-09-19 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (2.2 Å) Cite: The impact of cryosolution thermal contraction on proteins and protein crystals: volumes, conformation and order. Acta Crystallogr D Struct Biol, 74, 2018
6EAV	Crystallographic structure of the cyclic heptapeptide derived from the BTCI inhibitor bound to beta-trypsin in space group P 4(1) 2(1) 2 Descriptor: CALCIUM ION, CYS-THR-LYS, Cationic trypsin Authors: Fernandes, J.C, Valadares, N.F, Freitas, S.M, Barbosa, J.A.R.G. Deposit date: 2018-08-03 Release date: 2019-08-07 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (1.391 Å) Cite: Crystallographic structure of the cyclic heptapeptide derived from the BTCI inhibitor bound to beta-trypsin in space group P 4(1) 2(1) 2 To Be Published

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