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PDB: 5 results

1Y8O
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BU of 1y8o by Molmil
Crystal structure of the PDK3-L2 complex
Descriptor: ADENOSINE-5'-DIPHOSPHATE, DIHYDROLIPOIC ACID, Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, ...
Authors:Kato, M, Chuang, J.L, Wynn, R.M, Chuang, D.T.
Deposit date:2004-12-13
Release date:2005-05-24
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (2.48 Å)
Cite:Crystal structure of pyruvate dehydrogenase kinase 3 bound to lipoyl domain 2 of human pyruvate dehydrogenase complex.
Embo J., 24, 2005
2PNR
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BU of 2pnr by Molmil
Crystal Structure of the asymmetric Pdk3-l2 Complex
Descriptor: DIHYDROLIPOIC ACID, Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, [Pyruvate dehydrogenase [lipoamide]] kinase isozyme 3
Authors:Vassylyev, D.G, Steussy, C.N, Devedjiev, Y.
Deposit date:2007-04-25
Release date:2007-08-21
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Crystal Structure of an Asymmetric complex of Pyruvate Dehydrogenase Kinase 3 with Lipoyl domain 2 and its Biological Implications
J.Mol.Biol., 370, 2007
2Q8I
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BU of 2q8i by Molmil
Pyruvate dehydrogenase kinase isoform 3 in complex with antitumor drug radicicol
Descriptor: DIHYDROLIPOIC ACID, Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, GLYCEROL, ...
Authors:Kato, M, Li, J, Chuang, J.L, Chuang, D.T.
Deposit date:2007-06-10
Release date:2007-07-24
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Distinct Structural Mechanisms for Inhibition of Pyruvate Dehydrogenase Kinase Isoforms by AZD7545, Dichloroacetate, and Radicicol.
Structure, 15, 2007
1Y8N
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BU of 1y8n by Molmil
Crystal structure of the PDK3-L2 complex
Descriptor: DIHYDROLIPOIC ACID, Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, POTASSIUM ION, ...
Authors:Kato, M, Chuang, J.L, Wynn, R.M, Chuang, D.T.
Deposit date:2004-12-13
Release date:2005-05-24
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Crystal structure of pyruvate dehydrogenase kinase 3 bound to lipoyl domain 2 of human pyruvate dehydrogenase complex.
Embo J., 24, 2005
1Y8P
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BU of 1y8p by Molmil
Crystal structure of the PDK3-L2 complex
Descriptor: ADENOSINE-5'-TRIPHOSPHATE, DIHYDROLIPOIC ACID, Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, ...
Authors:Kato, M, Chuang, J.L, Wynn, R.M, Chuang, D.T.
Deposit date:2004-12-13
Release date:2005-05-24
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (2.63 Å)
Cite:Crystal structure of pyruvate dehydrogenase kinase 3 bound to lipoyl domain 2 of human pyruvate dehydrogenase complex.
Embo J., 24, 2005

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