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PDB: 2 results

8R37
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BU of 8r37 by Molmil
Klebsiella pneumoniae fosfomycin-resistance protein (FosAKP)
Descriptor: FOSFOMYCIN, FosA family fosfomycin resistance glutathione transferase, L(+)-TARTARIC ACID, ...
Authors:Papageorgiou, A.C, Varotsou, C, Labrou, N.E.
Deposit date:2023-11-08
Release date:2024-01-24
Method:X-RAY DIFFRACTION (1.48 Å)
Cite:Structural Studies of Klebsiella pneumoniae Fosfomycin-Resistance Protein and Its Application for the Development of an Optical Biosensor for Fosfomycin Determination.
Int J Mol Sci, 25, 2023
6C3U
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BU of 6c3u by Molmil
Crystal structure of Klebsiella pneumoniae fosfomycin resistance protein (FosAKP) with inhibitor (ANY2) bound
Descriptor: 3-bromo-6-(4-nitro-1H-pyrazol-3-yl)pyrazolo[1,5-a]pyrimidin-2(1H)-one, FosA family fosfomycin resistance glutathione transferase, GLYCEROL, ...
Authors:Klontz, E.H, Sundberg, E.J.
Deposit date:2018-01-10
Release date:2018-12-26
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Small-Molecule Inhibitor of FosA Expands Fosfomycin Activity to Multidrug-Resistant Gram-Negative Pathogens.
Antimicrob. Agents Chemother., 63, 2019

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