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PDB: 3 results

6W1M
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BU of 6w1m by Molmil
Cryo-EM structure of 5HT3A receptor in presence of Ondansetron
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(4-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 5-hydroxytryptamine receptor 3A, ...
Authors:Basak, S, Chakrapani, S.
Deposit date:2020-03-04
Release date:2021-01-13
Method:ELECTRON MICROSCOPY (3.06 Å)
Cite:High-resolution structures of multiple 5-HT 3A R-setron complexes reveal a novel mechanism of competitive inhibition.
Elife, 9, 2020
6W1Y
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BU of 6w1y by Molmil
Cryo-EM structure of 5HT3A receptor in presence of Palonosetron
Descriptor: (3~{a}~{S})-2-[(3~{S})-1-azabicyclo[2.2.2]octan-3-yl]-3~{a},4,5,6-tetrahydro-3~{H}-benzo[de]isoquinolin-1-one, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(4-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Basak, S, Chakrapani, S.
Deposit date:2020-03-04
Release date:2021-01-13
Method:ELECTRON MICROSCOPY (3.35 Å)
Cite:High-resolution structures of multiple 5-HT 3A R-setron complexes reveal a novel mechanism of competitive inhibition.
Elife, 9, 2020
6W1J
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BU of 6w1j by Molmil
Cryo-EM structure of 5HT3A receptor in presence of Alosetron
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(4-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 5-hydroxytryptamine receptor 3A, ...
Authors:Basak, S, Chakrapani, S.
Deposit date:2020-03-04
Release date:2021-01-13
Method:ELECTRON MICROSCOPY (2.92 Å)
Cite:High-resolution structures of multiple 5-HT 3A R-setron complexes reveal a novel mechanism of competitive inhibition.
Elife, 9, 2020

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