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PDB: 1 results

7AX4
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Human TYK2 pseudokinase domain (575-869) in complex with 5-(4-Fluoro-phenyl)-2-ureido-thiophene-3-carboxylic acid amide.
Descriptor: 2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamide, CALCIUM ION, Non-receptor tyrosine-protein kinase TYK2
Authors:Rowland, P.
Deposit date:2020-11-09
Release date:2021-04-14
Last modified:2024-05-15
Method:X-RAY DIFFRACTION (2.12 Å)
Cite:Reducing False Positives through the Application of Fluorescence Lifetime Technology: A Comparative Study Using TYK2 Kinase as a Model System.
SLAS Discov, 26, 2021

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