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PDB: 2 results

4YU9
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BU of 4yu9 by Molmil
Crystal Structure of double mutant Y115E Y117E human Glutaminyl Cyclase
Descriptor: 1,2-ETHANEDIOL, Glutaminyl-peptide cyclotransferase, SULFATE ION, ...
Authors:Di Pisa, F, Pozzi, C, Benvenuti, M, Mangani, S.
Deposit date:2015-03-18
Release date:2015-08-05
Last modified:2024-05-08
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:The soluble Y115E-Y117E variant of human glutaminyl cyclase is a valid target for X-ray and NMR screening of inhibitors against Alzheimer disease.
Acta Crystallogr.,Sect.F, 71, 2015
4YWY
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BU of 4ywy by Molmil
Crystal Structure of double mutant Y115E Y117E human Glutaminyl Cyclase in complex with inhibitor PBD-150
Descriptor: 1,2-ETHANEDIOL, 1-(3,4-dimethoxyphenyl)-3-[3-(1H-imidazol-1-yl)propyl]thiourea, CHLORIDE ION, ...
Authors:Di Pisa, F, Pozzi, C, Benvenuti, M, Mangani, S.
Deposit date:2015-03-21
Release date:2015-08-05
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:The soluble Y115E-Y117E variant of human glutaminyl cyclase is a valid target for X-ray and NMR screening of inhibitors against Alzheimer disease.
Acta Crystallogr.,Sect.F, 71, 2015

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