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PDB: 2 results

4Y85
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BU of 4y85 by Molmil
Crystal structure of COT kinase domain in complex with 5-(5-(1H-indol-3-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3,4-oxadiazol-2-amine
Descriptor: 5-[5-(1H-indol-3-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amine, Mitogen-activated protein kinase kinase kinase 8
Authors:Gutmann, S, Hinniger, A.
Deposit date:2015-02-16
Release date:2015-05-06
Last modified:2019-05-29
Method:X-RAY DIFFRACTION (2.33 Å)
Cite:The Crystal Structure of Cancer Osaka Thyroid Kinase Reveals an Unexpected Kinase Domain Fold.
J.Biol.Chem., 290, 2015
4Y83
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BU of 4y83 by Molmil
Crystal structure of COT kinase domain in complex with 5-(2-amino-5-(quinolin-3-yl)pyridin-3-yl)-1,3,4-oxadiazole-2(3H)-thione
Descriptor: 5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3H)-thione, Mitogen-activated protein kinase kinase kinase 8
Authors:Gutmann, S, Hinniger, A.
Deposit date:2015-02-16
Release date:2015-05-06
Last modified:2019-10-16
Method:X-RAY DIFFRACTION (2.89 Å)
Cite:The Crystal Structure of Cancer Osaka Thyroid Kinase Reveals an Unexpected Kinase Domain Fold.
J.Biol.Chem., 290, 2015

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