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PDB: 1 results

4FXY
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Crystal structure of rat neurolysin with bound pyrazolidin inhibitor
Descriptor: 1-{(2S)-1-[(3R)-3-(2-chlorophenyl)-2-(2-fluorophenyl)pyrazolidin-1-yl]-1-oxopropan-2-yl}-3-[(1R,3S,5R,7R)-tricyclo[3.3.1.1~3,7~]dec-2-yl]urea, Neurolysin, mitochondrial, ...
Authors:Rodgers, D.W, Hines, C.S.
Deposit date:2012-07-03
Release date:2013-11-13
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Allosteric inhibition of the neuropeptidase neurolysin.
J.Biol.Chem., 289, 2014

223790

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