English
日本語
简体中文
繁體中文
한국어
✖
Menu
RCSB PDB
PDBe
BMRB
Adv. Search
Search help
PDB: 6 results
4M14
Crystal structure of ITK in complex with compound 9 [4-(carbamoylamino)-1-[7-(propan-2-yloxy)naphthalen-1-yl]-1H-pyrazole-3-carboxamide]
Descriptor:
4-(carbamoylamino)-1-[7-(propan-2-yloxy)naphthalen-1-yl]-1H-pyrazole-3-carboxamide, Tyrosine-protein kinase ITK/TSK
Authors:
Han, S
,
Caspers, N.L.
Deposit date:
2013-08-02
Release date:
2014-04-02
Last modified:
2024-02-28
Method:
X-RAY DIFFRACTION (1.55 Å)
Cite:
Selectively targeting an inactive conformation of interleukin-2-inducible T-cell kinase by allosteric inhibitors.
Biochem.J., 460, 2014
4M15
Crystal structure of ITK in complex with compound 9 [4-(carbamoylamino)-1-[7-(propan-2-yloxy)naphthalen-1-yl]-1H-pyrazole-3-carboxamide] and ADP
Descriptor:
4-(carbamoylamino)-1-[7-(propan-2-yloxy)naphthalen-1-yl]-1H-pyrazole-3-carboxamide, ADENOSINE-5'-DIPHOSPHATE, Tyrosine-protein kinase ITK/TSK
Authors:
Han, S
,
Caspers, N.L.
Deposit date:
2013-08-02
Release date:
2014-04-02
Last modified:
2024-02-28
Method:
X-RAY DIFFRACTION (1.52 Å)
Cite:
Selectively targeting an inactive conformation of interleukin-2-inducible T-cell kinase by allosteric inhibitors.
Biochem.J., 460, 2014
4M0Y
Crystal structure of ITK in complex with compound 1 [4-(carbamoylamino)-1-(naphthalen-1-yl)-1H-pyrazole-3-carboxamide]
Descriptor:
4-(carbamoylamino)-1-(naphthalen-1-yl)-1H-pyrazole-3-carboxamide, Tyrosine-protein kinase ITK/TSK
Authors:
Han, S
,
Caspers, N.L.
Deposit date:
2013-08-02
Release date:
2014-04-02
Last modified:
2024-02-28
Method:
X-RAY DIFFRACTION (1.7 Å)
Cite:
Selectively targeting an inactive conformation of interleukin-2-inducible T-cell kinase by allosteric inhibitors.
Biochem.J., 460, 2014
4M13
Crystal structure of ITK in complex with compound 8 [4-(carbamoylamino)-1-(7-propoxynaphthalen-1-yl)-1H-pyrazole-3-carboxamide]
Descriptor:
4-(carbamoylamino)-1-(7-propoxynaphthalen-1-yl)-1H-pyrazole-3-carboxamide, Tyrosine-protein kinase ITK/TSK
Authors:
Han, S
,
Caspers, N.L.
Deposit date:
2013-08-02
Release date:
2014-04-02
Last modified:
2024-02-28
Method:
X-RAY DIFFRACTION (1.85 Å)
Cite:
Selectively targeting an inactive conformation of interleukin-2-inducible T-cell kinase by allosteric inhibitors.
Biochem.J., 460, 2014
4M12
Crystal structure of ITK in complex with compound 7 [4-(carbamoylamino)-1-(7-ethoxynaphthalen-1-yl)-1H-pyrazole-3-carboxamide]
Descriptor:
4-(carbamoylamino)-1-(7-ethoxynaphthalen-1-yl)-1H-pyrazole-3-carboxamide, Tyrosine-protein kinase ITK/TSK
Authors:
Han, S
,
Caspers, N.L.
Deposit date:
2013-08-02
Release date:
2014-04-02
Last modified:
2024-02-28
Method:
X-RAY DIFFRACTION (2.15 Å)
Cite:
Selectively targeting an inactive conformation of interleukin-2-inducible T-cell kinase by allosteric inhibitors.
Biochem.J., 460, 2014
4M0Z
Crystal structure of ITK in complex with compound 5 {4-(carbamoylamino)-1-(7-methoxynaphthalen-1-yl)-1H-pyrazole-3-carboxamide}
Descriptor:
4-(carbamoylamino)-1-(7-methoxynaphthalen-1-yl)-1H-pyrazole-3-carboxamide, Tyrosine-protein kinase ITK/TSK
Authors:
Han, S
,
Caspers, N.L.
Deposit date:
2013-08-02
Release date:
2014-04-02
Last modified:
2024-02-28
Method:
X-RAY DIFFRACTION (2 Å)
Cite:
Selectively targeting an inactive conformation of interleukin-2-inducible T-cell kinase by allosteric inhibitors.
Biochem.J., 460, 2014
Home
Top Page
Statistics
Help
FAQ
Contact Us
Cite Us / Terms and Conditions
Links
Settings
Data deposition (OneDep)
Help
Deposition to PDB, EMDB or BMRB
Download
Download PDB archive / snapshot archive
Standard format
PDBx/mmCIF Resources
Format Conversion
PDBx/mmCIF editor
Quick links
Help
non-PDB format compatible
Group Depositions
Chemical Component entries
Latest entries
Search services
Help
Search PDB (PDBj Mine)
Search PDBj RDB
Chemie search
Search BMRB
Sequence-Navigator
DASH
EM Navigator
Omokage search
SeSAW
wwPDB/RDF
RDF Portal
Status search
Molecular Viewers
Help
jV: Graphic Viewer
Molmil: WebGL Mol. Viewer
Services & Softwares
Help
Yorodumi
ASH
MAFFTash
NMRToolBox
gmfit
CRNPRED
Spanner
SFAS
HOMCOS
Derived databases
Help
eF-site
eF-seek
eF-surf
ProMode Elastic
hGTOP
Educational service
Help
eProtS
Molecule of the Month
Previous workshop
Games
Papermodels
About PDBj
Help
Publications
Newsletters / Public Relations Resources
PDBj Members
PDBj Advisory Committee
Privacy Policy
218853
PDB entries from 2024-04-24