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PDB: 2 results
5VK0
Crystal structure of human MDM2 in complex with a 12-mer lysine-cysteine side chain dithiocarbamate stapled peptide inhibitor PMI
Descriptor:
CHLORIDE ION, E3 ubiquitin-protein ligase Mdm2, Lysine-cysteine side chain dithiocarbamate stapled peptide inhibitor PMI
Authors:
Tolbert, W.D
,
Gohain, N
,
Pazgier, M.
Deposit date:
2017-04-20
Release date:
2018-04-25
Last modified:
2023-10-04
Method:
X-RAY DIFFRACTION (1.8 Å)
Cite:
Dithiocarbamate-inspired side chain stapling chemistry for peptide drug design.
Chem Sci, 10, 2019
5VK1
Crystal structure of human MDM4 in complex with a 12-mer lysine-cysteine side chain dithiocarbamate stapled peptide inhibitor PMI
Descriptor:
Lysine-cysteine side chain dithiocarbamate stapled peptide inhibitor PMI, Protein Mdm4
Authors:
Tolbert, W.D
,
Gohain, N
,
Pazgier, M.
Deposit date:
2017-04-20
Release date:
2018-04-25
Last modified:
2023-10-04
Method:
X-RAY DIFFRACTION (2.69 Å)
Cite:
Dithiocarbamate-inspired side chain stapling chemistry for peptide drug design.
Chem Sci, 10, 2019
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PDB entries from 2024-04-24