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PDB: 1 results

5TTZ
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BU of 5ttz by Molmil
Crystal structure of Grp94 bound to isoform-selective inhibitor methyl 2-(2-(1-(4-bromobenzyl)-1H-imidazol-2-yl)ethyl)-3-chloro-4,6-dihydroxybenzoate
Descriptor: 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, DI(HYDROXYETHYL)ETHER, Endoplasmin, ...
Authors:Lieberman, R.L, Huard, D.J.E.
Deposit date:2016-11-04
Release date:2018-01-10
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.707 Å)
Cite:Isoform-selective Hsp90 inhibition rescues model of hereditary open-angle glaucoma.
Sci Rep, 7, 2017

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