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PDB: 1 results

6GY0
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BU of 6gy0 by Molmil
mPI3Kd IN COMPLEX WITH AZ3
Descriptor: Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform, ~{N}-[4-methyl-5-(1-oxidanylidene-7-sulfamoyl-isoindol-5-yl)-1,3-thiazol-2-yl]ethanamide
Authors:Petersen, J.
Deposit date:2018-06-27
Release date:2019-02-06
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (2.55 Å)
Cite:A class of highly selective inhibitors bind to an active state of PI3K gamma.
Nat.Chem.Biol., 15, 2019

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