Loading
PDBj
MenuPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 1 results

8A7I
DownloadVisualize
BU of 8a7i by Molmil
Crystal structure of BRD9 bromodomain in complex with compound EA-89
Descriptor: Bromodomain-containing protein 9, ~{N}-[1,1-bis(oxidanylidene)thian-4-yl]-7-[3-methyl-1-(piperidin-4-ylmethyl)indol-5-yl]-4-oxidanylidene-5-propyl-thieno[3,2-c]pyridine-2-carboxamide
Authors:Faller, M, Zink, F.
Deposit date:2022-06-21
Release date:2022-08-10
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.76 Å)
Cite:BRD9 degraders as chemosensitizers in acute leukemia and multiple myeloma.
Blood Cancer J, 12, 2022

238895

PDB entries from 2025-07-16

PDB statisticsPDBj update infoContact PDBjnumon