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8A7I
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BU of 8a7i by Molmil
Crystal structure of BRD9 bromodomain in complex with compound EA-89
Descriptor: Bromodomain-containing protein 9, ~{N}-[1,1-bis(oxidanylidene)thian-4-yl]-7-[3-methyl-1-(piperidin-4-ylmethyl)indol-5-yl]-4-oxidanylidene-5-propyl-thieno[3,2-c]pyridine-2-carboxamide
Authors:Faller, M, Zink, F.
Deposit date:2022-06-21
Release date:2022-08-10
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.76 Å)
Cite:BRD9 degraders as chemosensitizers in acute leukemia and multiple myeloma.
Blood Cancer J, 12, 2022

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PDB entries from 2024-07-17

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