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PDB: 3 results

3MVH
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BU of 3mvh by Molmil
Crystal structure of Akt-1-inhibitor complexes
Descriptor: GSK3-beta peptide, MANGANESE (II) ION, N-{[(3S)-3-amino-1-(5-ethyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamide, ...
Authors:Pandit, J.
Deposit date:2010-05-04
Release date:2010-06-02
Last modified:2021-10-06
Method:X-RAY DIFFRACTION (2.01 Å)
Cite:Design of selective, ATP-competitive inhibitors of Akt.
J.Med.Chem., 53, 2010
3MV5
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BU of 3mv5 by Molmil
Crystal structure of Akt-1-inhibitor complexes
Descriptor: (3R)-1-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine, GSK3-beta peptide, MANGANESE (II) ION, ...
Authors:Pandit, J.
Deposit date:2010-05-03
Release date:2010-06-02
Last modified:2021-10-06
Method:X-RAY DIFFRACTION (2.47 Å)
Cite:Design of selective, ATP-competitive inhibitors of Akt.
J.Med.Chem., 53, 2010
3MVJ
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BU of 3mvj by Molmil
Human cyclic AMP-dependent protein kinase PKA inhibitor complex
Descriptor: (3R)-1-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine, cAMP-dependent protein kinase catalytic subunit alpha, cAMP-dependent protein kinase inhibitor alpha
Authors:Pandit, J, Vajdos, F.
Deposit date:2010-05-04
Release date:2010-06-02
Last modified:2017-11-08
Method:X-RAY DIFFRACTION (2.49 Å)
Cite:Design of selective, ATP-competitive inhibitors of Akt.
J.Med.Chem., 53, 2010

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