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PDB: 1 results

5LXM
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BU of 5lxm by Molmil
Crystal structure of Aurora-A bound to a hydrocarbon-stapled proteomimetic of TPX2
Descriptor: 1-ETHOXY-2-(2-ETHOXYETHOXY)ETHANE, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ADENOSINE-5'-DIPHOSPHATE, ...
Authors:McIntyre, P.J, Bayliss, R.
Deposit date:2016-09-22
Release date:2016-11-02
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.08 Å)
Cite:A TPX2 Proteomimetic Has Enhanced Affinity for Aurora-A Due to Hydrocarbon Stapling of a Helix.
ACS Chem. Biol., 11, 2016

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