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PDB: 2 results

7AQT
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BU of 7aqt by Molmil
NMR2 structure of BRD4-BD2 in complex with iBET-762
Descriptor: 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide, Bromodomain-containing protein 4
Authors:Orts, J, Torres, F, Milbradt, A.G, Walser, R.
Deposit date:2020-10-23
Release date:2022-03-02
Last modified:2022-04-27
Method:SOLUTION NMR
Cite:NMR Molecular Replacement Provides New Insights into Binding Modes to Bromodomains of BRD4 and TRIM24.
J.Med.Chem., 65, 2022
7B9X
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BU of 7b9x by Molmil
NMR2 structure of TRIM24-BD in complex with a precursor of IACS-9571
Descriptor: N-{6-[3-(4-Aminobutoxy)-5-propoxyphenoxy]-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl}-3,4-dimethoxybenzene-1-sulfonamide, Transcription intermediary factor 1-alpha
Authors:Orts, J, Torres, F, Milbradt, A.G, Walser, R.
Deposit date:2020-12-14
Release date:2022-01-12
Last modified:2022-04-27
Method:SOLUTION NMR
Cite:NMR Molecular Replacement Provides New Insights into Binding Modes to Bromodomains of BRD4 and TRIM24.
J.Med.Chem., 65, 2022

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