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PDB: 1 results

7OVY
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BU of 7ovy by Molmil
Crystal structure of a dimeric based inhibitor JG34 in complex with the MMP-12 catalytic domain
Descriptor: 1,2-ETHANEDIOL, CALCIUM ION, Macrophage metalloelastase, ...
Authors:Ciccone, L, Rossello, A, Vera, L, Nuti, E, Stura, E.A.
Deposit date:2021-06-15
Release date:2021-10-27
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.24 Å)
Cite:Discovery of Dimeric Arylsulfonamides as Potent ADAM8 Inhibitors.
Acs Med.Chem.Lett., 12, 2021

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