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7P4S
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BROMODOMAIN OF HUMAN TAF1 (2) WITH naphthyridinone compound
Descriptor: 8-[[1-(3-azanylpropyl)piperidin-4-yl]amino]-5-[5-(hydroxymethyl)pyridin-3-yl]-3-methyl-1~{H}-1,7-naphthyridin-2-one, Isoform 2a of Transcription initiation factor TFIID subunit 1
Authors:Chung, C.
Deposit date:2021-07-13
Release date:2021-10-13
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.17 Å)
Cite:Optimization of Naphthyridones into Selective TATA-Binding Protein Associated Factor 1 (TAF1) Bromodomain Inhibitors.
Acs Med.Chem.Lett., 12, 2021

221371

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