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PDB: 1 results

6I8Z
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BU of 6i8z by Molmil
Crystal structure of PTK2 in complex with BI-4464.
Descriptor: 3-methoxy-~{N}-(1-methylpiperidin-1-ium-4-yl)-4-[[4-[(3-oxidanylidene-1,2-dihydroinden-4-yl)oxy]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide, Focal adhesion kinase 1
Authors:Bader, G, Zoephel, A.
Deposit date:2018-11-21
Release date:2019-02-20
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (1.99 Å)
Cite:Highly Selective PTK2 Proteolysis Targeting Chimeras to Probe Focal Adhesion Kinase Scaffolding Functions.
J.Med.Chem., 62, 2019

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