8WQO
 
 | | Crystal structure of BRD4-BD1 bound with DI106 | | Descriptor: | (3~{R})-6-[[4-(3,5-dimethyl-1~{H}-pyrazol-4-yl)pyrimidin-2-yl]amino]-1,3-dimethyl-4-propan-2-yl-3~{H}-quinoxalin-2-one, Isoform C of Bromodomain-containing protein 4 | | Authors: | Cao, D, Xiong, B. | | Deposit date: | 2023-10-12 | | Release date: | 2024-07-24 | | Last modified: | 2025-02-19 | | Method: | X-RAY DIFFRACTION (1.13 Å) | | Cite: | Structure-Based Rational Design and Evaluation of BET-Aurora Kinase Dual-Inhibitors for Treatment of Cancers.
J.Med.Chem., 68, 2025
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