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PDB: 1 results

8A3Q
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BU of 8a3q by Molmil
Human Plasma Kallekrein in complex with 14W
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, Plasma kallikrein, ...
Authors:McEwan, P.A.
Deposit date:2022-06-08
Release date:2022-11-02
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.801 Å)
Cite:Sebetralstat (KVD900): A Potent and Selective Small Molecule Plasma Kallikrein Inhibitor Featuring a Novel P1 Group as a Potential Oral On-Demand Treatment for Hereditary Angioedema.
J.Med.Chem., 65, 2022

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