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PDB: 2 results

7JYO
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BU of 7jyo by Molmil
JAK2 JH2 in complex with JAK064
Descriptor: 3-({4-amino-6-[(4-cyanophenyl)amino]-1,3,5-triazin-2-yl}oxy)benzoic acid, GLYCEROL, Tyrosine-protein kinase JAK2
Authors:Puleo, D.E, Krimmer, S.G, Newton, A.S, Schlessinger, J, Jorgensen, W.L.
Deposit date:2020-08-31
Release date:2021-07-14
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.16127229 Å)
Cite:Indoloxytriazines as binding molecules for the JAK2 JH2 pseudokinase domain and its V617F variant
Tetrahedron Lett., 77, 2021
7JYQ
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BU of 7jyq by Molmil
JAK2 JH2 in complex with JAK020
Descriptor: GLYCEROL, N~2~-(4-fluorophenyl)-6-{[(5-{[(oxolan-2-yl)methyl]amino}-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-1,3,5-triazine-2,4-diamine, Tyrosine-protein kinase JAK2
Authors:Puleo, D.E, Krimmer, S.G, Newton, A.S, Schlessinger, J, Jorgensen, W.L.
Deposit date:2020-08-31
Release date:2021-07-14
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (1.85941613 Å)
Cite:Indoloxytriazines as binding molecules for the JAK2 JH2 pseudokinase domain and its V617F variant
Tetrahedron Lett., 77, 2021

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