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PDB: 1 results

7N9G
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BU of 7n9g by Molmil
Crystal structure of the Abl 1b Kinase domain in complex with Dasatinib and Imatinib
Descriptor: 4-(4-METHYL-PIPERAZIN-1-YLMETHYL)-N-[4-METHYL-3-(4-PYRIDIN-3-YL-PYRIMIDIN-2-YLAMINO)-PHENYL]-BENZAMIDE, N-(2-CHLORO-6-METHYLPHENYL)-2-({6-[4-(2-HYDROXYETHYL)PIPERAZIN-1-YL]-2-METHYLPYRIMIDIN-4-YL}AMINO)-1,3-THIAZOLE-5-CARBOXAMIDE, PHOSPHATE ION, ...
Authors:Miller, D.J, Xie, T.
Deposit date:2021-06-17
Release date:2022-04-27
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Imatinib can act as an Allosteric Activator of Abl Kinase.
J.Mol.Biol., 434, 2022

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