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PDB: 2 results

7R5B
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BU of 7r5b by Molmil
Crystal structure of BRD4(1) in complex with the inhibitor MPM2
Descriptor: (R,R)-2,3-BUTANEDIOL, 1-(3-aminophenyl)-3-methyl-5,6,7,8-tetrahydro-2~{H}-cyclohepta[c]pyrrol-4-one, Bromodomain-containing protein 4, ...
Authors:Huegle, M.
Deposit date:2022-02-10
Release date:2023-02-08
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.77 Å)
Cite:A novel pan-selective bromodomain inhibitor for epigenetic drug design
Eur.J.Med.Chem., 249, 2023
7B1T
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BU of 7b1t by Molmil
Crystal structure of BRD4(1) in complex with the inhibitor MPM6
Descriptor: 3-(5-azanyl-2-chloranyl-phenyl)-1-methyl-4,7-dihydro-2~{H}-cyclohepta[c]pyrrol-8-one, Bromodomain-containing protein 4, DIMETHYL SULFOXIDE
Authors:Huegle, M.
Deposit date:2020-11-25
Release date:2022-06-08
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.92 Å)
Cite:A novel pan-selective bromodomain inhibitor for epigenetic drug design.
Eur.J.Med.Chem., 249, 2023

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PDB entries from 2024-10-16

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