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PDB: 2 results

5V9O
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BU of 5v9o by Molmil
KRAS G12C inhibitor
Descriptor: GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
Authors:Westover, K, Lu, J.
Deposit date:2017-03-23
Release date:2017-08-23
Last modified:2024-10-30
Method:X-RAY DIFFRACTION (1.56 Å)
Cite:Potent and Selective Covalent Quinazoline Inhibitors of KRAS G12C.
Cell Chem Biol, 24, 2017
5V9L
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BU of 5v9l by Molmil
KRAS G12C in bound to quinazoline based switch II pocket (SWIIP) binder
Descriptor: GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
Authors:Westover, K, Lu, J.
Deposit date:2017-03-23
Release date:2017-08-23
Last modified:2024-10-30
Method:X-RAY DIFFRACTION (1.981 Å)
Cite:Potent and Selective Covalent Quinazoline Inhibitors of KRAS G12C.
Cell Chem Biol, 24, 2017

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