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7LQ1
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HUMAN PI3KDELTA IN COMPLEX WITH COMPOUND 28
Descriptor: CHLORIDE ION, N-(5-(6-(2-((2S,6R)-2,6-dimethylmorpholino)pyridin-4-yl)-1-oxoisoindolin-4-yl)-2-methoxypyridin-3-yl)methanesulfonamide, Phosphatidylinositol 3-kinase regulatory subunit alpha, ...
Authors:Lesburg, C.A, Augustin, M.
Deposit date:2021-02-12
Release date:2022-02-16
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (2.96 Å)
Cite:Discovery of a new series of PI3K-delta inhibitors from Virtual Screening.
Bioorg.Med.Chem.Lett., 42, 2021

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